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Cat. No. Product Name Target Signaling Pathways
TP1051 Protein Kinase C Peptide Substrate

PRKCE,Peptide Epsilon,PKCε

Protein Kinase C Peptide Substrate targets specific cell spacers ina manner that is dependent on second messengers and specific adaptor proteins in response to extracellular signals that activate g protein-coupled receptors, tyrosine Kinase receptors, or
T35827 Epsilon-V1-2

PKCε Inhibitor Peptide,Protein Kinase Cɛ Inhibitor Peptide,ɛV1-2

Protein kinase C (PKC ) is a calcium-independent, phospholipid- and diacylglycerol-dependent serine/threonine kinase involved in diverse signaling pathways, including those involved in neuronal signaling, cytoskeletal function, and inflammation.[1] PKC inhibitor peptide is a synthetic peptide corresponding to an amino acid sequence found in the amino terminal C2 domain of most mammalian forms of PKC .[2] It selectively and reversibly inhibits the translocation of PKC to intracellular membrane...
T80511 PKCε inhibitor peptide,myristoylated

Myr‐PKCɛ-

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Myristoylated PKCε inhibitor peptide(Myr-PKCε-)是一种与肉豆蔻酸偶联、具有细胞渗透性的PKCε蛋白激酶Cε亚型特异性肽抑制剂,它能够降低人脐静脉内皮细胞(HUVECs)的一氧化氮(NO)释放。
T82451 Epsilon-polylysine

ε-Polylysine,ε-PL

Epsilon-polylysine 是由特定细菌产生的抗菌肽,主要用作食品和饮料的防腐剂。它能有效抑制各类微生物如细菌、酵母菌和霉菌的生长。该化合物因其热稳定性、耐酸性和广谱抗菌活性,成为理想的食品添加剂。
T80249 Epsilon-V1-2, Cys-conjugated

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Epsilon-V1-2, Cys-conjugated 是 εPKC 特异性抑制剂,通过阻断 εPKC 与 εRACK 锚定蛋白之间的相互作用,抑制 εPKC 易位及 MARCKS 磷酸化,从而表现生物活性。该肽将半胱氨酸残基接到 C 末端,以形成与载体蛋白的 SS 键。当序列 N 末端为谷氨酰胺 (Q) 或谷氨酸 (E) 时,肽可自发生成焦谷氨酰 (pGlu)。Q或E到pGlu的转化属于自然过程,并且pGlu的疏水性γ-内酰胺环对提高肽对胃肠道蛋白酶的稳定性起关键作用。在 HPLC 分析中,焦谷氨酰肽作为肽纯度的一部分进行检测,视为这类肽的典型子集。

化合物

Protein Kinase C Peptide Substrate
Cat.No: TP1051
Synonym: PRKCE,Peptide Epsilon,PKCε
Target:
Epsilon-V1-2
Cat.No: T35827
Synonym: PKCε Inhibitor Peptide,Protein Kinase Cɛ Inhibitor Peptide,ɛV1-2
Target:
PKCε inhibitor peptide,myristoylated
Cat.No: T80511
Synonym: Myr‐PKCɛ-
Target: PKC
Epsilon-polylysine
Cat.No: T82451
Synonym: ε-Polylysine,ε-PL
Target:
Epsilon-V1-2, Cys-conjugated
Cat.No: T80249
Synonym:
Target: PKC
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