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Cat. No. Product Name Target Signaling Pathways
T13842 PROTAC IRAK4 degrader-1

Others Others
PROTAC IRAK4 degrader-1 is a degrader of PROTAC interleukin-1 receptor-associated kinase 4 (IRAK4).
T7755 Thalidomide 4-fluoride

E3 ligase Ligand 4,2-(2,6-二氧代-哌啶-3-基)-4-氟基-异吲哚-1,3-二酮

IRAK; Ligand for E3 Ligase Immunology/Inflammation; NF-κB; PROTAC
Thalidomide 4-fluoride (E3 ligase Ligand 4) 是一种基于 Thalidomide 的 Cereblon 配体,可用于募集 CRBN 蛋白。它能够利用 linker 与 IRAK4 靶蛋白配体连接,得到 PROTAC IRAK4 degrader-1
T81378 PROTAC IRAK4 ligand-3

PROTACs PROTAC
PROTACIRAK4 ligand-3 为 PROTACIRAK4 degrader-7 配体,适用于癌症研究领域。
T79097 PROTAC IRAK4 degrader-8

IRAK Immunology/Inflammation; NF-κB
PROTAC-IRAK4分解剂-8(化合物2)是针对IRAK4设计的PROTAC,表现出15.5 nM的IC50值。
T74411 PROTAC IRAK4 degrader-7

PROTACIRAK4 degrader-7 (Compound I-417) 是一种具有口服活性的 PROTACIRAK4降解剂,具有抗肿瘤效果。
T39903 PROTAC IRAK4 degrader-6

PROTAC IRAK4 degrader-6

PROTAC IRAK4 degrader-6 is a potent Cereblon-based compound designed to degrade interleukin-1 receptor-associated kinase 4 (IRAK4).
T39901 PROTAC IRAK4 degrader-4

PROTAC IRAK4 degrader-4

PROTAC IRAK4 degrader-4 (US20190192668A1, compound I-127) is a Cereblon-based PROTAC specifically designed to target and degrade interleukin-1 receptor-associated kinase 4 (IRAK4).
T17388 AM-Imidazole-PA-Boc

Others Others
AM-Imidazole-PA-Boc is an alkyl chain-derived PROTAC linker utilized for the synthesis of PROTAC IRAK4 degrader-1[1].
T74062 PROTAC IRAK4 degrader-2

PROTACIRAK4 degrader-2 (Compound 9) 是一种 PROTACIRAK4降解剂,在外周血单个核细胞 (PBMC) 中,降解 IRAK4,DC50为 151 nM。PROTACIRAK4 Degrader-2 在 PBMC 细胞中诱导 IRAK4蛋白水平降低,DC50为 36 nM。PROTACIRAK4 degrader-2 还抑制 PBMC 中多种细胞因子释放。

化合物

PROTAC IRAK4 degrader-1
Cat.No: T13842
Synonym:
Target: Others
Thalidomide 4-fluoride
Cat.No: T7755
Synonym: E3 ligase Ligand 4,2-(2,6-二氧代-哌啶-3-基)-4-氟基-异吲哚-1,3-二酮
Target: IRAK, Ligand for E3 Ligase
PROTAC IRAK4 ligand-3
Cat.No: T81378
Synonym:
Target: PROTACs
PROTAC IRAK4 degrader-8
Cat.No: T79097
Synonym:
Target: IRAK
PROTAC IRAK4 degrader-7
Cat.No: T74411
Synonym:
Target:
PROTAC IRAK4 degrader-6
Cat.No: T39903
Synonym: PROTAC IRAK4 degrader-6
Target:
PROTAC IRAK4 degrader-4
Cat.No: T39901
Synonym: PROTAC IRAK4 degrader-4
Target:
AM-Imidazole-PA-Boc
Cat.No: T17388
Synonym:
Target: Others
PROTAC IRAK4 degrader-2
Cat.No: T74062
Synonym:
Target:
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