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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T60169 |
BLU0588
|
Others | Others |
BLU0588是一种选择性的PRKACA 抑制剂。BLU0588以1nM 的 IC50 抑制PRKACA 催化活性。 | |||
T60170 |
BLU2864
|
Others | Others |
BLU2864 是一种具有口服活性的、高选择性的、ATP 竞争性的 PRKACA 抑制剂 ,IC50值为0.3 nM。BLU2864 具有抗肿瘤活性,具有用于癌症和多囊肾的研究潜力。 | |||
T63041 | DS01080522 | ||
DS01080522 是一种 PRKACA 的抑制剂。DS01080522 对 PRKACA 激酶的活性 (IC50: 0.8 nM) 以及 CREB 磷酸化 (IC50: 66 nM) 具有抑制作用。DS0108052 能够用于研究癌症。 | |||
T62676 | DS89002333 | ||
DS89002333 是一种强效的、口服具有活力的 PRKACA 抑制剂 (IC50: 0.3 nM)。DS89002333 在表达 DNAJB1-PRKACA 融合基因的 FL-HCC 患者源性异种移植模型中具有良好的抗肿瘤作用。DS89002333 能够用于研究纤维化肝细胞癌 (FL-HCC)。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPK-00677 |
PKA/PRKACA Protein, Canine, Recombinant (His)
PKA C alpha,PKACA,PPNAD4,PKA C α,PKA C-α,PKA C-alpha,PRK... |
Canine | E. coli |
The cAMP-dependent protein kinase PKA is a well-characterized member of the serine-threonine protein AGC kinase family and is the effector kinase of cAMP signaling. As such, PKA is involved in the control of a wide variety of cellular processes including metabolism, cell growth, gene expression and apoptosis. cAMP-dependent PKA signaling pathways play important roles during infection and virulence of various pathogens. Since fluxes in cAMP are involved in multiple intracellular functions, a vari... |