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Targets Recommended: Others

12

抑制剂 & 化合物

1

天然产物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T12772 (RS)-PPG

Others Others
(RS)-PPG is a potent and selective group III mGluRs agonist(EC50s of 5.2 μM, 4.7 μM, 185 μM, and 0.2 μM for hmGluR4a, hmGluR6, hmGluR7b, and hmGluR8a, respectively),with neuroprotective and anticonvulsive activity.
T38714 Boc-NH-PPG2

Boc-NH-PPG2

Boc-NH-PPG2 is a alkyl/ether-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
TF0060 DPPG

DPPG 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0060,CAS号为 200880-41-7。
T10880 CPPG

(RS)-CPPG

Others Others
CPPG is a potent antagonist of group II/III mGlu receptors. CPPG exhibits some selectivity (approximately 20 fold) for group III (IC50: 2.2 nM) over group II (IC50: 46.2 nM) mGlu receptors in the rat cerebral cortex.
T74477 m7GpppGmpG ammonium

m7GpppGmpG ammonium 是一种三核苷酸 5′ 端帽类似物。m7GpppGmpG 对 RNA 的加帽率为 86%。
T82485 ELAAWCRWGFLLALLPPGIAG

ELAAWCRWGFLLALLPPGIAG (P5) 是源自大鼠HER2/neu蛋白的21个氨基酸长肽(氨基酸5-25)。此肽可诱导携带HER2阳性肿瘤小鼠中的细胞毒性T淋巴细胞(CTL)反应。
T83687 Mca-RPPGFSAFK(Dnp)-OH TFA

(7-methoxycoumarin-4-yl)acetyl-Arg-Pro-Pro-Gly-Phe-Ser-Ala-Phe-Lys(2,4-dinitrophenyl)-OH

Mca-RPPGFSAFK(Dnp)-OH 是 endothelin-converting enzyme-1 (ECE-1) 的一种荧光底物。当 ECE-1 切割该底物时,会释放 7-methoxycoumarin-4-acetyl (Mca),其荧光可以用来量化 ECE-1 的活性。Mca 的激发/发射峰值分别为 328/420 nm。
T32617 L-DPPG

L-Dipalmitoylphosphatidylglycerol

L-DPPG is a bioactive chemical.
T74475 m7GpppGpG

m7GpppGpG 是 M7GpppNpG 三核苷酸帽类似物的一种寡核苷酸。它能够防止 5'-外切核酸酶过早的降解作用,并能够募集前 mRNA 剪接、mRNA 转运以及蛋白质生物合成启动所需的蛋白质。
T38212 MPPG

MPPG 是一种有选择性的 L-AP4 敏感受体拮抗剂(kD=9.2 μM)。
T74476 m7GpppGmpG

m7GpppGmpG 是一种三核苷酸 5′ 端帽类似物。m7GpppGmpG 对 RNA 的加帽率为 86%。
T82484 ELAAWCRWGFLLALLPPGIAG TFA

ELAAWCRWGFLLALLPPGIAG TFA (P5) 是由大鼠HER2/neu蛋白衍生的21个氨基酸长的肽段(氨基酸序号5至25)。该化合物在携带HER2阳性肿瘤的小鼠模型中,能够诱发细胞毒性T淋巴细胞(CTL)的反应。

化合物

(RS)-PPG
Cat.No: T12772
Synonym:
Target: Others
Boc-NH-PPG2
Cat.No: T38714
Synonym: Boc-NH-PPG2
Target:
DPPG
Cat.No: TF0060
Synonym:
Target:
CPPG
Cat.No: T10880
Synonym: (RS)-CPPG
Target: Others
m7GpppGmpG ammonium
Cat.No: T74477
Synonym:
Target:
ELAAWCRWGFLLALLPPGIAG
Cat.No: T82485
Synonym:
Target:
Mca-RPPGFSAFK(Dnp)-OH TFA
Cat.No: T83687
Synonym: (7-methoxycoumarin-4-yl)acetyl-Arg-Pro-Pro-Gly-Phe-Ser-Ala-Phe-Lys(2,4-dinitrophenyl)-OH
Target:
L-DPPG
Cat.No: T32617
Synonym: L-Dipalmitoylphosphatidylglycerol
Target:
m7GpppGpG
Cat.No: T74475
Synonym:
Target:
MPPG
Cat.No: T38212
Synonym:
Target:
m7GpppGmpG
Cat.No: T74476
Synonym:
Target:
ELAAWCRWGFLLALLPPGIAG TFA
Cat.No: T82484
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T83673 4-Hydroxyphenylpropionylglycine

Phloretylglycine,4-hydroxy PPG,Phloretic Acid Glycine Conjugate

4-Hydroxyphenylpropionylglycine是一种由条件必需氨基酸酪氨酸代谢形成的代谢产物。通过芳香族氨基酸转氨酶、酪氨酸转氨酶以及肠道微生物作用后,结合甘氨酸共轭生成。此外,4-Hydroxyphenylpropionylglycine也是酚类化合物phloretin的代谢产物。

天然产物

4-Hydroxyphenylpropionylglycine
Cat.No: T83673
Synonym: Phloretylglycine,4-hydroxy PPG,Phloretic Acid Glycine Conjugate
Target:
Cat. No. Product Name Species Expression System
TMPY-03436 Serglycin Protein, Human, Recombinant (His)

PRG1,PPG,serglycin,PRG

Human HEK293 Cells
Serglycin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.1 kDa and the accession number is AAA60179.1.
TMPY-02373 Serglycin Protein, Human, Recombinant (His & Myc)

PRG,serglycin,PRG1,PPG

Human HEK293 Cells
Serglycin Protein, Human, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with His and Myc tag. The predicted molecular weight is 17.3 kDa and the accession number is AAA60179.1.

重组蛋白

Serglycin Protein, Human, Recombinant (His)
Cat.No: TMPY-03436
Species: Human
Expression System: HEK293 Cells
Serglycin Protein, Human, Recombinant (His & Myc)
Cat.No: TMPY-02373
Species: Human
Expression System: HEK293 Cells
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