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Cat. No. Product Name Target Signaling Pathways
T12455 PI3K/HDAC-IN-1

PI3K PI3K/Akt/mTOR signaling
PI3K/HDAC-IN-1 is a potent PI3K and HDAC dual inhibitor(IC50s of 8.1 nM and 1.4 nM, respectively).
T62545 HDAC-IN-43

HDAC-IN-43 是一种强效的 HDAC 1/3/6 抑制剂,对 HDAC 1HDAC 3 和 HDAC 6 的 IC50 值分别为 82 nM、45 nM 和 24 nM。HDAC-IN-43 是一种弱的 PI3K/mTOR 抑制剂,对 PI3K 和 mTOR 的 IC50 值分别为 3.6 μM 和 3.7 μM。HDAC-IN-43 具有广谱的抗增殖效果。
T81499 PH14

PI3K PI3K/Akt/mTOR signaling
PH14,作为一种PI3K/HDAC双重抑制剂,对PI3Kα和HDAC3表现出强效抑制能力,其IC50值分别为20.3 nM 和24.5 nM 。该化合物不仅具备抗增殖特性,还能有效诱导Jeko-1细胞走向凋亡,是研究癌症(例如淋巴瘤)的有力工具。
T36421 Immuno-Oncology Screening Library

The Immuno-Oncology Screening Library consists of 2 plates and contains more than 90 cancer and immunology-associated compounds in a 96-well Matrix tube rack format as 10 mM stock solutions in DMSO. This library includes a variety of immuno-oncology target modulators, including but not limited to, adenosine, CCR, CXCR, and TLR agonists and antagonists, BTK, PI3K, VEGFR, and BRAF inhibitors, PD-1/PDL-1 interaction inhibitors, and HDAC inhibitors. Please review the product insert for a full list ...

化合物

PI3K/HDAC-IN-1
Cat.No: T12455
Synonym:
Target: PI3K
HDAC-IN-43
Cat.No: T62545
Synonym:
Target:
PH14
Cat.No: T81499
Synonym:
Target: PI3K
Immuno-Oncology Screening Library
Cat.No: T36421
Synonym:
Target:
TargetMol Loading
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