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Cat. No. Product Name Target Signaling Pathways
T4221 PF-06260933

PF-6260933,PF 6260933,PF6260933

MAPK MAPK
PF-06260933 是一种具有高度选择性及口服有活性的MAP4K4小分子抑制剂,在激酶实验中IC50为 3.7 nM,在细胞实验中IC50为 160 nM。
T36016 PF 06260933 dihydrochloride

MAP4K4 (HGK) inhibitor (IC50 = 140 nM). Also inhibits MINK and TNIK (IC50 values are 8 and 13 nM, respectively). Improves fasting hyperglycemia in mice. Orally active. Ammirati et al (2015) Discovery of an in vivo tool to establish proof-of-concept for MAP4K4-based antidiabetic treatment. ACS Med.Chem.Lett. 6 1128 PMID:26617966
T33945 PF-06260933 HCl

PF06260933 dihydrochloride,PF-06260933 dihydrochloride,PF 06260933 dihydrochloride

PF-06260933 Dihydrochloride is a MAP4K4 (HGK) inhibitor (IC50 = 140 nM). It can improve the fasting hyperglycemia in mice. In addition, it inhibited Mink and Tnik (IC50 values of 8 and 13 nM, respectively).

化合物

PF-06260933
Cat.No: T4221
Synonym: PF-6260933,PF 6260933,PF6260933
Target: MAPK
PF 06260933 dihydrochloride
Cat.No: T36016
Synonym:
Target:
PF-06260933 HCl
Cat.No: T33945
Synonym: PF06260933 dihydrochloride,PF-06260933 dihydrochloride,PF 06260933 dihydrochloride
Target:
TargetMol Loading
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