Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12344L1 |
OTS186935 FA
OTS186935 FA(2093400-18-9 Free base) |
Histone Methyltransferase | Chromatin/Epigenetic |
OTS186935 FA 是一种蛋白甲基转移酶 SUV39H2 抑制剂。OTS186935 FA在 MDA-MB-231 乳腺癌细胞和 A549 肺癌细胞中抑制肿瘤的生长。 | |||
T63654 | OTS186935 hydrochloride | ||
OTS186935 hydrochloride 是蛋白甲基转移酶 SUV39H2 的有效抑制剂 (IC50: 6.49 nM)。OTS186935 hydrochloride 在小鼠异种移植模型中,能够明显抑制肿瘤生长,且没有明显毒性。OTS193320 hydrochloride 能够调节癌细胞中 γ-H2AX 的产生。 | |||
T12344 |
OTS186935
|
Others | Others |
OTS186935 is a inhibitor of protein methyltransferase SUV39H2(IC50 of 6.49 nM). | |||
T12344L |
OTS186935 trihydrochloride
|
Others | Others |
OTS186935 trihydrochloride is a protein methyltransferase inhibitor of SUV39H2(IC50 of 6.49 nM). |