Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T31877 |
Freselestat
ONO-PO 736,ONO-6818,ONO 6818,ONO6818 |
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Freselestat (ONO-6818) is a potent neutrophil elastase inhibitor that significantly reduces the production of interleukin 8 and C5B-9. Freselestat reduces inflammatory mediators during simulated cardiopulmonary bypass. | |||
T62846 | Freselestat quarterhydrate | ||
Freselestat quarterhydrate (ONO-6818 quarterhydrate) 是一种有效的、口服具有活力的嗜中性粒细胞弹性蛋白酶 (neutrophil elastase) 抑制剂 (Ki: 12.2 nM)。Freselestat quarterhydrate 对其他蛋白酶(例如胰蛋白酶,蛋白酶3,胰弹性蛋白酶,凝血酶,纤溶酶,胶原酶,组织蛋白酶G 和鼠巨噬细胞弹性蛋白酶)的活性低 100 倍以上,表现出有效的抗炎作用。 |