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Cat. No. | Product Name | Target | Signaling Pathways |
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T7769 |
Nonapeptide-1
Met-Pro-D-Phe-Arg-D-Trp-Phe-Lys-Pro-Val-,九胜肽-1,Melanostatine™ 5 |
Others | Others |
Nonapeptide-1 (Melanostatine™ 5) 可以抑制黑色素的合成,这使得它对治疗某些皮肤病很感兴趣。 | |||
TP1101 |
Nonapeptide-1 acetate salt (158563-45-2 free base)
Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt |
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) 是一种肽激素,是一种有效的 α-黑色素细胞刺激素 (α-MSH) 拮抗剂,IC50 为 11 nM。 | |||
T75715 |
Nonapeptide-1 acetate salt
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Nonapeptide-1 (Melanostatine-5) acetate salt,一种多肽类激素,是 MC1R 选择性拮抗剂 (Ki: 40 nM)。 Nonapeptide-1 acetate salt 是一种竞争性的α-MSH 拮抗剂,可有效抑制黑素细胞中 α-MSH 诱导的细胞内 cAMP 和黑素体扩散 (IC50分别为 2.5 nM 和 11 nM)。 Nonapeptide-1 acetate salt 抑制黑色素合成,可用于研究皮肤色素沉着和肾上腺类固醇生成的调节、皮肤癌。 | |||
TP1819L |
Substance P 1-9 aceate
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Neurotensin Receptor | GPCR/G Protein |
Substance P 1-9 aceate 是九肽,可减少豚鼠回肠和膀胱对 P 物质的失活。 | |||
TP1496L |
p5 Ligand for Dnak and DnaJ acetate
p5 Ligand for Dnak and DnaJ acetate(209518-24-1 free base) |
HSP | Cytoskeletal Signaling; Metabolism |
p5 Ligand for Dnak and DnaJ acetate(209518-24-1 free base) 是一种九肽。它是 DnaK(大肠杆菌 Hsp70)和 DnaJ(大肠杆菌 Hsp40)的高亲和力配体。 | |||
T37664 |
Emideltide (acetate)
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Emideltide, also known as delta sleep-inducing peptide (DSIP), is a synthetic nonapeptide sedative.1 | |||
T80962 |
TPNQRQNVC
LRH-1 peptide |
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TPNQRQNVC为HLA-B0702的九肽抗原决定簇,能激活CD8+ T细胞的免疫响应。 | |||
T80540 |
TCMCB07
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Melanocortin Receptor | GPCR/G Protein; Neuroscience |
TCMCB07为环状九肽,是具有口服活性及脑渗透性的黑皮质素受体4 (MC4R) 拮抗剂,在恶病质中具有关键作用。 | |||
TP1435 |
Chemerin-9 (149-157) TFA(676367-27-4 free base)
Chemerin-9 (149-157) (TFA) |
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Chemerin-9 (149-157) TFA, the nonapeptide (149)YFPGQFAFS(157) (chemerin-9), corresponding to the C terminus of processed chemerin, retains most of the activity of the full-size protein, with regard to agonism toward the chemerinR[1]. | |||
T37890 |
GLP-1(28-36)amide
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GLP-1(28-36)amide, a C-terminal nonapeptide derived from the cleavage of GLP-1 by neutral endopeptidase (NEP), is a significant product. It functions as an antioxidant and primarily targets the mitochondrion, where it effectively inhibits mitochondrial permeability transition (MPT). This compound exhibits anti-diabetic properties and demonstrates cardioprotection effects[1]. | |||
TP1819 |
Substance P (1-9)
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Substance P (1-9) is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder. Subtance P is responsible for a number of excitatory effects on both central and peripheral neurons. | |||
T80911 |
Tyrosinase (192-200), human mouse
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Tyrosinase(192-200), human mouse 为九肽化合物,能被HLA-B44分子所识别的细胞溶解T细胞(CTL)所识别,常用于黑色素瘤相关癌症研究。 | |||
T80541 |
TCMCB07 TFA
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Melanocortin Receptor | GPCR/G Protein; Neuroscience |
TCMCB07 TFA为一环状九肽,属口服活性及脑渗透性黑皮质素受体4 (MC4R) 拮抗剂,于恶病质中扮演关键角色。 | |||
T76191 |
GLP-1(28-36)amide TFA
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GLP-1(28-36)amide TFA,为GLP-1 C-端九肽段,主要通过中性内肽酶(NEP)裂解GLP-1生成。该化合物作为一种抗氧化剂,能靶向线粒体,抑制线粒体通透性转变(MPT),显示出抗糖尿病和心脏保护的功效。 | |||
T75799 |
Hemopressin(human, mouse) TFA
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Cannabinoid Receptor | GPCR/G Protein |
Hemopressin TFA,一种衍生自血红蛋白α1链的九肽,最初自大鼠脑匀浆分离。作为口服活性且选择性的CB1大麻素受体反向激动剂,Hemopressin TFA在炎性疼痛模型中具有抗伤害感受效应。 | |||
T76550 |
CooP
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CooP为一种针对线性胶质母细胞瘤的九肽,与胶质母细胞瘤细胞及其相关血管系统中的乳腺来源生长抑制剂/脂肪酸结合蛋白3 (FABP3) 发生结合。该化合物主要应用于化学疗法和多种纳米粒子的靶向递送。 | |||
T75798 | Hemopressin(rat) TFA | ||
Hemopressin(rat) TFA,一种衍生自α1-珠蛋白九肽,最初分离自大鼠脑匀浆。该化合物通过口服能有效选择性地作为CB1大麻素受体的反向激动剂,并在炎性疼痛模型中表现出抗伤害感受活性。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T73954 | Leucinostatin (mixture of A&B) | ||
Leucinostatin (mixture of A&B) 是来自Paecilomyces lilacinus 的九肽类复合物,具有抗生素活性。 |