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Cat. No. Product Name Target Signaling Pathways
T1524 Nilotinib

尼洛替尼,尼罗替尼,Tasigna,AMN107

Bcr-Abl; Autophagy Angiogenesis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Nilotinib (AMN107) 是一种 Bcr-Abl 酪氨酸激酶抑制剂,具有抗肿瘤活性。
T2147 Nilotinib monohydrochloride monohydrate

Nilotinib (monohydrochloride monohydrate),尼洛替尼盐酸盐一水合物,AMN107 (monohydrochloride monohydrate),尼罗替尼中间体

Bcr-Abl; Autophagy Angiogenesis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Nilotinib monohydrochloride monohydrate (Nilotinib (monohydrochloride monohydrate)) 是酪氨酸酶抑制剂,有效抑制 BCR-ABL 及其突变体。
T22378 Nilotinib hydrochloride

AMN-107 HCl

Bcr-Abl; Autophagy Angiogenesis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Nilotinib hydrochloride(AMN-107 HCl) 是一种可口服的 Bcr-Abl 酪氨酸激酶抑制,具有抗肿瘤活性,可用于调节神经炎症和认知障碍,可用于研究慢性骨髓性白血病。
T68338 Nilotinib hydrochloride dihydrate

Nilotinib hydrochloride dihydrate is a small-molecule tyrosine kinase inhibitor approved for the treatment of imatinib-resistant chronic myelogenous leukemia.
T19035 Nilotinib Acid

Others Others
Nilotinib Acid, an analog of Nilotinib, is usually used as a fluorescent probe or labeled chemical.
T71068 Nilotinib dihydrochloride dihydrate

Nilotinib dihydrochloride dihydrate is a small-molecule tyrosine kinase inhibitor approved for the treatment of imatinib-resistant chronic myelogenous leukemia.
T12224 Nilotinib-d6

AMN107 D6

Others Others
Nilotinib D6 is a deuterium labeled Nilotinib which is an orally available inhibitor of Bcr-Abl tyrosine kinase ,and with antineoplastic activity.
T71144 Nilotinib N-oxide

Nilotinib N-oxide is a small-molecule tyrosine kinase inhibitor approved for the treatment of imatinib-resistant chronic myelogenous leukemia.
T71142 Tebuconazole-d9

Tebuconazole-d9 is intended for use as an internal standard for the quantification of tebuconazole by GC- or LC-MS. Tebuconazole is a triazole fungicide that is active against both seed and foliar fungi. It inhibits 14α-demethylase isolated from U. maydis and S. bicolor with IC50 values of 0.05 and 0.16 nM, respectively. It inhibits the androgenic effect of the androgen receptor agonist DHT (IC20 = 2.89 µM) and is cytotoxic (EC20 = 38.9 µM) in an MDA-kb2 assay. Tebuconazole (50 and 100 mg/kg per...
T71066 Cidofovir sodium

Cidofovir sodium is the salt form of Cidofovir, a Cytomegalovirus Nucleoside Analog DNA Polymerase Inhibitor that is an injectable antiviral medication primarily used as a treatment for cytomegalovirus (CMV) retinitis in people with AIDS. The mechanism of action of cidofovir is as a DNA Polymerase Inhibitor. The chemical classification of cidofovir anhydrous is Nucleoside Analog.
T71581 SGX393

SGX393 is an inhibitor of the CML mutant Bcr-AblT315I, thereby preempting in vitro resistance when combined with nilotinib or dasatinib.

化合物

Nilotinib
Cat.No: T1524
Synonym: 尼洛替尼,尼罗替尼,Tasigna,AMN107
Target: Bcr-Abl, Autophagy
Nilotinib monohydrochloride monohydrate
Cat.No: T2147
Synonym: Nilotinib (monohydrochloride monohydrate),尼洛替尼盐酸盐一水合物,AMN107 (monohydrochloride monohydrate),尼罗替尼中间体
Target: Bcr-Abl, Autophagy
Nilotinib hydrochloride
Cat.No: T22378
Synonym: AMN-107 HCl
Target: Bcr-Abl, Autophagy
Nilotinib hydrochloride dihydrate
Cat.No: T68338
Synonym:
Target:
Nilotinib Acid
Cat.No: T19035
Synonym:
Target: Others
Nilotinib dihydrochloride dihydrate
Cat.No: T71068
Synonym:
Target:
Nilotinib-d6
Cat.No: T12224
Synonym: AMN107 D6
Target: Others
Nilotinib N-oxide
Cat.No: T71144
Synonym:
Target:
Tebuconazole-d9
Cat.No: T71142
Synonym:
Target:
Cidofovir sodium
Cat.No: T71066
Synonym:
Target:
SGX393
Cat.No: T71581
Synonym:
Target:
TargetMol Loading
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