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Cat. No. Product Name Target Signaling Pathways
T2325 Neratinib

HKI-272,来那替尼

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Neratinib (HKI-272) 是一种口服的、不可逆的酪氨酸激酶抑制剂,对 HER2 和 EGFR 的 IC50值分别为 59 和 92 nM。
T67385 Neratinib maleate

HKI-272 maleate

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Neratinib maleate (HKI-272 maleate) 是一种不可逆且具有口服活性和高选择性的 HER2 和 EGFR 抑制剂,IC50 值分别为 59 nM 和 92 nM。Neratinib maleate具有抗肿瘤活性,可用于治疗消化系统疾病、呼吸系统疾病、泌尿生殖系统疾病和皮肤和肌肉骨骼疾病,可用于研究乳腺癌和前列腺癌。
T71387 Neratinib maleate monohydrate

Neratinib maleate monohydrate is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity.
T70829 Neratinib pyridine N-oxide

Neratinib pyridine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity.
T70830 Neratinib dimethylamine N-oxide

Neratinib dimethylamine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity.
T70828 HBY-793

HBY-793 is an HIV-1 proteinase inhibitor.
T70827 MDL-102234

MDL-102234 is an adenosine A1 receptor antagonist.

化合物

Neratinib
Cat.No: T2325
Synonym: HKI-272,来那替尼
Target: EGFR, HER
Neratinib maleate
Cat.No: T67385
Synonym: HKI-272 maleate
Target: EGFR, HER
Neratinib maleate monohydrate
Cat.No: T71387
Synonym:
Target:
Neratinib pyridine N-oxide
Cat.No: T70829
Synonym:
Target:
Neratinib dimethylamine N-oxide
Cat.No: T70830
Synonym:
Target:
HBY-793
Cat.No: T70828
Synonym:
Target:
MDL-102234
Cat.No: T70827
Synonym:
Target:
TargetMol Loading
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