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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T8312 Derenofylline

Adenosine Receptor GPCR/G Protein; Neuroscience
Derenofylline 是一个有选择性的、具有口服活性的腺苷A1受体的拮抗剂,可抑制心肌纤维化,降低蛋白尿,对腺苷A1、A3和A2A 受体的Ki 值分别为 1、200 和 398 nM。
T69966 Roxadustat-d5

Roxadustat-d5 is intended for use as an internal standard for the quantification of roxadustat by GC- or LC-MS. Roxadustat is an inhibitor of hypoxia-inducible factor prolyl hydroxylase (HIF-PH; IC50s = 1.4, 1.26, and 1.32 µM for HIF-PH1, HIF-PH2, and HIF-PH3, respectively). It is selective for HIF-PH over other 2-oxoglutarate-dependent dioxygenases, including lysine-specific demethylase 5A (KDM5A), KDM5B, -5C, -5D, and -6B (IC50s = >100 µM for all). Roxadustat (10-200 µM) stabilizes HIF-1α and ...

化合物

Derenofylline
Cat.No: T8312
Synonym:
Target: Adenosine Receptor
Roxadustat-d5
Cat.No: T69966
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3033 Deoxycorticosterone acetate

醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮

Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。

天然产物

Deoxycorticosterone acetate
Cat.No: T3033
Synonym: 醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮
Target: Glucocorticoid Receptor, Endogenous Metabolite, Adrenergic Receptor
TargetMol Loading
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