Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1827 |
Buparlisib
BKM120,布帕尼西,NVP-BKM120 |
Apoptosis; PI3K | Apoptosis; PI3K/Akt/mTOR signaling |
Buparlisib (BKM120) 是一种具有口服生物利用度的泛 I 类 PI3K 特异性口服抑制剂,对p110α/p110β/p110δ/p110γ的IC50分别为 52 nM/166 nM/116 nM/262 nM。 | |||
T16365 |
Buparlisib Hydrochloride
NVP-BKM120 Hydrochloride,BKM120 Hydrochloride |
Others | Others |
Buparlisib Hydrochloride is an inhibitor of pan-class I PI3K (IC50: 52 nM/166 nM/116 nM/262 nM for p110α/p110β/p110δ/p110γ, respectively). |