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Cat. No. Product Name Target Signaling Pathways
T5394 Prulifloxacin

AF 3012,Pruvel,NM441,普卢利沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Prulifloxacin (NM441) 是一种口服有效的氟喹诺酮抗生素 ,对革兰氏阳性和阴性细菌具有广泛活性。它是噻唑喹啉羧酸衍生物 Ulifloxacin 的前药。它有潜力用于下尿路感染和慢性支气管炎。
T21325 TAK-441

TAK441

Hedgehog/Smoothened GPCR/G Protein; Stem Cells
TAK-441 是一种具有口服活性的 Hedgehog 信号抑制剂 (IC50 = 4.4 nM),具有有效的抗肿瘤活性。 TAK-441 抑制转录因子 Gli1 mRNA 表达和肿瘤生长。
TP1013 N-CBZ-Phe-Arg-AMC

Z-FR-AMC

N-CBZ-Phe-Arg-AMC (Z-FR-AMC) is a substrate for serine proteases, including cathepsins, kallikrein and plasmin. Absorption/emission of substrate = 330/390 nm (weak fluorescence); absorption/emission of end product (AMC) = 342/441 nm (strong fluorescence).
TP1562 F1324

F1324 is a potent, high affinity peptidic inhibitor of B cell lymphoma 6 (BCL6) with an IC50 of 1 nM. F1324 exhibits binding t1/2 value of 441 s and has strong inhibition activity against BCL6 PPI.
T37338 N-3-oxo-pentanoyl-L-Homoserine lactone

N-3-oxo-pentanoyl-L-Homoserine lactone is a chain-shortened derivative of the bacterial quorum sensing signaling molecule N-3-oxo-octanoyl-L-homoserine lactone .1It inhibits binding of the autoinducer N-3-oxo-hexanoyl homoserine lactone toE. colicontaining the transcription factor LuxR when used at a concentration of 230 nM.2It acts as an autoinducer to activate theV. fischeriluminescence system inE. coliwhen used at concentrations ranging from 20 to 200 nM. 1.Chhabra, S.R., Stead, P., Bainton, ...

化合物

Prulifloxacin
Cat.No: T5394
Synonym: AF 3012,Pruvel,NM441,普卢利沙星
Target: Topoisomerase, Antibacterial, Antibiotic
TAK-441
Cat.No: T21325
Synonym: TAK441
Target: Hedgehog/Smoothened
N-CBZ-Phe-Arg-AMC
Cat.No: TP1013
Synonym: Z-FR-AMC
Target:
F1324
Cat.No: TP1562
Synonym:
Target:
N-3-oxo-pentanoyl-L-Homoserine lactone
Cat.No: T37338
Synonym:
Target:
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