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Cat. No. Product Name Target Signaling Pathways
T6812L Cyclo(-RGDfK) TFA

Integrin Cytoskeletal Signaling
Cyclo(-RGDfK) TFA 是一种选择性整合素αvβ3的有效抑制剂,其IC50值为 0.94 nM。它通过与细胞表面的 αvβ3 整合素结合,特异性靶向肿瘤微血管和癌细胞。
T6812 Cyclo(-RGDfK)

Cyclo (-RGDfK)

Integrin Cytoskeletal Signaling
Cyclo(-RGDfK) (Cyclo (-RGDfK)) 是一种选择性整合素αvβ3的有效抑制剂,IC50值为 0.94 nM。它通过与细胞表面的 αvβ3 整合素结合,特异性靶向肿瘤微血管和癌细胞。
T2064 Semaxinib

司马沙尼,SU5416

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
Semaxinib (SU5416) 是一种选择性的 VEGFR(Flk-1/KDR) 抑制剂,其 IC50=1.23 μM。
T68400 STA-9584

STA-9584 is a potent vascular disrupting agent, which exhibits potent antitumor activity by selectively targeting microvasculature at both the center and periphery of tumors. In vitro, 2-methoxy-5-(5-(3,4,5-trimethoxyphenyl)isoxazol-4-yl)aniline (STA-9122) (active metabolite of STA-9584 ) displayed increased potency relative to other tubulin-binding agents and was highly cytotoxic to tumor cells. STA-9584 induced significant tumor regressions in prostate and breast xenograft models in vivo and, ...

化合物

Cyclo(-RGDfK) TFA
Cat.No: T6812L
Synonym:
Target: Integrin
Cyclo(-RGDfK)
Cat.No: T6812
Synonym: Cyclo (-RGDfK)
Target: Integrin
Semaxinib
Cat.No: T2064
Synonym: 司马沙尼,SU5416
Target: VEGFR
STA-9584
Cat.No: T68400
Synonym:
Target:
TargetMol Loading
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