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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T19717 Cyclo-L-Trp-L-Trp

Antifungal Microbiology/Virology
Cyclo-L-Trp-L-Trp 是一种广谱抗真菌剂。它还诱导组蛋白的高度乙酰化。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。

化合物

Cyclo-L-Trp-L-Trp
Cat.No: T19717
Synonym:
Target: Antifungal
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
TN3080 5,6,7-Trimethoxycoumarin

P450; Antifection Metabolism; Microbiology/Virology
5,6,7-Trimethoxycoumarin shows moderate inhibitory activity against Micrococcus luteus, it also displays an intermediate cytotoxic effects against brine shrimp larvae. 5,6,7-Trimethoxycoumarin can improve gastroprotective effects, and it has low toxicity
TN2625 14-Deoxycoleon U

Antifection Microbiology/Virology
14-Deoxycoleon U has anti-termitic activity, it is highly active against both wood-decay fungi. 14-Deoxycoleon U shows antibacterial activity against the Gram-positive bacteria Staphylococcus aureus, Staphylococcus epidermidis, Enterococcus faecalis, and

天然产物

Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
5,6,7-Trimethoxycoumarin
Cat.No: TN3080
Synonym:
Target: P450, Antifection
14-Deoxycoleon U
Cat.No: TN2625
Synonym:
Target: Antifection
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