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6

抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T5954 Methyldopa hydrate

L-甲基多巴,Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate

Dopamine Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Methyldopa hydrate (MK-351 hydrate) 是一种前药,在中枢神经系统中被代谢成 α-Methylepinephrine。它是一种 α-肾上腺素能激动剂,对α2-adrenergic receptors 有选择性。
T15701 Methyldopa hydrochloride

L-(-)-α-Methyldopa hydrochloride,MK-351 hydrochloride

Others Others
L-(-)-α-Methyldopa hydrochloride is an alpha-adrenergic agonist psychoactive drug. It is used as a sympatholytic or antihypertensive. Methyldopa has a dual mechanism of action. It is a competitive inhibitor of the enzyme DOPA decarboxylase, which converts
T69105 Methyldopa anhydrous

Methyldopa anhydrous is a Central alpha-2 Adrenergic Agonist. The mechanism of action of methyldopa anhydrous is as an Adrenergic alpha2-Agonist.
T20133 Methyldopate hydrochloride

Aldomet Ester hydrochloride,Aldomet,Methyldopate HCl,Methyldopa ethyl ester hydrochloride

Methyldopate HCl is an agent of antihypertensive.
T36206 Methyldopate

Methyldopate is an ethyl ester prodrug form of methyldopa , a dopamine decarboxylase inhibitor that has antihypertensive activity in vitro and in vivo., Formulations containing methyldopate have been used in the treatment of hypertension.
T60241 N-Methyldopamine hydrochloride

N-Methyldopamine hydrochloride 是肾上腺素在肾上腺髓质中的前体。N-Methyldopamine hydrochloride 是多巴胺 (DA) 的修饰物,并保留了对 DA1 受体 (DA1 receptor) 的激动剂活性。N-Methyldopamine hydrochloride 具有普遍的表面包覆和利用表面儿茶酚进行二次反应的能力。N-Methyldopamine hydrochloride 可用于心力衰竭的研究。

化合物

Methyldopa hydrate
Cat.No: T5954
Synonym: L-甲基多巴,Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate
Target: Dopamine Receptor, Adrenergic Receptor
Methyldopa hydrochloride
Cat.No: T15701
Synonym: L-(-)-α-Methyldopa hydrochloride,MK-351 hydrochloride
Target: Others
Methyldopa anhydrous
Cat.No: T69105
Synonym:
Target:
Methyldopate hydrochloride
Cat.No: T20133
Synonym: Aldomet Ester hydrochloride,Aldomet,Methyldopate HCl,Methyldopa ethyl ester hydrochloride
Target:
Methyldopate
Cat.No: T36206
Synonym:
Target:
N-Methyldopamine hydrochloride
Cat.No: T60241
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0505 Methyldopa

L-(-)-α-Methyldopa,MK-351,甲基多巴

Dopamine Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
L-(-)-α-Methyldopa (MK-351) 是一种前药,在中枢神经系统中被代谢成 α-Methylepinephrine。它是 α-肾上腺素能激动剂,对 α2- adrenergic receptors 有选择性。

天然产物

Methyldopa
Cat.No: T0505
Synonym: L-(-)-α-Methyldopa,MK-351,甲基多巴
Target: Dopamine Receptor, Adrenergic Receptor
TargetMol Loading
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