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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T7211 Tyr-Gly-Gly-Phe-Met-OH

Methionine enkephalin,蛋氨酸脑啡肽,Met-Enkephalin,[MET5]脑啡肽

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin) 是天然存在的内源性阿片肽、metenkephalin 和 zeta-和 delta-阿片受体激动剂的合成形式,是 mu-阿片受体激动剂,具有潜在的镇痛、神经调节、免疫调节、抗炎、抗肿瘤作用以及镇痛、抗抑郁和胃肠运动调节活性。
T31632 Enkephalin-met, acetaldehyde-

Methionine-enkephalin, acetaldehyde,Met-enkephalin, acetaldehyde,Acetaldehyde-met-enkephalin

Enkephalin-met, a naturally occurring opioid peptide used to regulate the growth of human colon cancer, can be used as an effective negative regulator of human gastrointestinal cancer and may suggest pathways for tumor etiology, progression, treatment and
T31634 [Des-Tyr1]-Met-Enkephalin

Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-

Enkephalin-met, des-tyr(1)- ccauses retrograde amnesia in rats.
TP1254 [Met5]-Enkephalin, amide TFA

5-Methionine-enkephalin amide (TFA)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) (60117-17-1 free base) 是一种 δ 阿片受体激动剂以及推定的 ζ (zeta) opioid 受体。
T31633 Enkephalin-met, ala(2)-

Dalmee,DAMET,Met-enkephalin, ala(2)-

Enkephalin-met, ala(2)- is a synthetic analog of methionine enkephalin.
T31635 Enkephalin-met, lys(6)-

Met-enk-L,6-Lys-met-enkephalin

Enkephalin-met, lys(6)- is an opioid hexapeptide found in adrenal medulla.
T31636 Enkephalin-met, tyr-O-sulfate

METOS,Met-enkephalin, tyr-O-sulfate-,Tyr-O-sulfate-met-enkephalin

Enkephalin-met, tyr-O-sulfate is a opioid peptide.
TP1255 [Met5]-Enkephalin, amide

5-Methionine-enkephalin amide

[Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.Met-enkephalin circulates in several forms, some of which may be derived from proteins other than proenkephalin A, and plasma levels of both free n
T2208 Bacitracin Zinc

杆菌肽锌,Bacitracin zinc salt,Zinc bacitracin

c-Met/HGFR; Antibacterial; Antibiotic Microbiology/Virology; Tyrosine Kinase/Adaptors
Bacitracin Zinc 是 C55-异戊二烯焦磷酸酯的去磷酸化干扰物,可抑制 Met-enkephalin 中 Tyr 的裂解,IC50为10 μM。
T32019 Guanyl-damme

Guanyl damme

Guanyl-damme is an analog of stable met-enkephalin.
T20332 Bam 12P

Bam12P,Bam-12P

Bam 12P is a Pro-Met-enkephalin precursor that is isolated from the bovine adrenal medulla.
T25804L Metkephamid acetate

Lilly 127623,LY127623,LY-127623,LY 127623

Metkephamid acetate is a synthetic opioid pentapeptide and derivative of [Met]enkephalin. It shows as a potent agonist of the δ- and μ-opioid receptors with roughly equipotent affinity, and also has similarly high affinity as well as subtype-selectivity f
T81817 Met-Arg-Phe-Ala

Met-Arg-Phe-Ala为一种肽类化合物,同时作为脑啡肽生成内肽酶(EGE)的有效竞争性抑制剂,应用于神经系统疾病的研究。
T25804 Metkephamid

Metkefamida

Metkephamid is a synthetic opioid pentapeptide and derivative of [Met]enkephalin. It shows as a potent agonist of the δ- and μ-opioid receptors with roughly equipotent affinity, and also has similarly high affinity as well as subtype-selectivity for the κ
TP1914 BAM(8-22)

BAM (8-22)

Endogenous peptide fragment that is a potent agonist for MRGPRX1 (EC50 values are 8 - 150 nM); first isolated from bovine adrenal medulla. Unlike BAM 22P , does not contain the met-enkephalin motif therefore displays no affinity for opioid receptors.

化合物

Tyr-Gly-Gly-Phe-Met-OH
Cat.No: T7211
Synonym: Methionine enkephalin,蛋氨酸脑啡肽,Met-Enkephalin,[MET5]脑啡肽
Target: Opioid Receptor
Enkephalin-met, acetaldehyde-
Cat.No: T31632
Synonym: Methionine-enkephalin, acetaldehyde,Met-enkephalin, acetaldehyde,Acetaldehyde-met-enkephalin
Target:
[Des-Tyr1]-Met-Enkephalin
Cat.No: T31634
Synonym: Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-
Target:
[Met5]-Enkephalin, amide TFA
Cat.No: TP1254
Synonym: 5-Methionine-enkephalin amide (TFA)
Target: Opioid Receptor
Enkephalin-met, ala(2)-
Cat.No: T31633
Synonym: Dalmee,DAMET,Met-enkephalin, ala(2)-
Target:
Enkephalin-met, lys(6)-
Cat.No: T31635
Synonym: Met-enk-L,6-Lys-met-enkephalin
Target:
Enkephalin-met, tyr-O-sulfate
Cat.No: T31636
Synonym: METOS,Met-enkephalin, tyr-O-sulfate-,Tyr-O-sulfate-met-enkephalin
Target:
[Met5]-Enkephalin, amide
Cat.No: TP1255
Synonym: 5-Methionine-enkephalin amide
Target:
Bacitracin Zinc
Cat.No: T2208
Synonym: 杆菌肽锌,Bacitracin zinc salt,Zinc bacitracin
Target: c-Met/HGFR, Antibacterial, Antibiotic
Guanyl-damme
Cat.No: T32019
Synonym: Guanyl damme
Target:
Bam 12P
Cat.No: T20332
Synonym: Bam12P,Bam-12P
Target:
Metkephamid acetate
Cat.No: T25804L
Synonym: Lilly 127623,LY127623,LY-127623,LY 127623
Target:
Met-Arg-Phe-Ala
Cat.No: T81817
Synonym:
Target:
Metkephamid
Cat.No: T25804
Synonym: Metkefamida
Target:
BAM(8-22)
Cat.No: TP1914
Synonym: BAM (8-22)
Target:
Cat. No. Product Name Target Signaling Pathways
T81816 Met-Enkephalin-Arg-Phe

Met-Enkephalin-Arg-Phe 是一种天然七肽,具有镇痛活性。

天然产物

Met-Enkephalin-Arg-Phe
Cat.No: T81816
Synonym:
Target:
TargetMol Loading
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