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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0503 Meglumine

Meglumin,Methylglucamin,葡甲胺,葡萄糖甲胺,Methylglucamine

Others Others
Meglumine (Meglumin) 是一种氨基糖,来源于山梨糖醇。其中常在药物中用作赋形剂,并与碘代化合物葡甲胺和碘帕胺葡甲胺等造影剂中的碘化化合物一起使用。
T8173 Delafloxacin meglumine

ABT492 meglumine,德拉沙星葡甲胺,WQ-3034 meglumine,RX-3341 meglumine

Antibacterial; Antibiotic Microbiology/Virology
Delafloxacin meglumine (RX-3341 meglumine) 是一种广谱氟喹诺酮类抗生素。Delafloxacin 对耐药性的金黄色葡萄球菌,肺炎克雷伯菌和肺炎链球菌有活性。
T1209 Flunixin meglumine

Banamine,Finadyne,Flunixin meglumin,氟尼辛葡甲胺

COX Immunology/Inflammation; Neuroscience
Flunixin meglumine (Banamine) 是一种环氧合酶抑制剂,具有抗炎和解热活性。
T7582 tafamidis meglumine

Fx-1006A,他发米帝司甲葡胺

Others Others
Tafamidis meglumine (Fx-1006A) 是transthyretin (TTR)的选择性稳定剂,对野生型 WT-TTR 和突变型同源四聚体 V30M-TTR,V122I-TTR 的活性相当,EC50值为 2.7-3.2 μM。它能够阻碍淀粉样蛋白的生成。
T20637 Diatrizoate meglumine

Reno,Renografin,Renovist,泛影葡胺,Hypaque,Renocal,Sinografin

Others Others
Diatrizoate meglumine (Renocal) 是泛影酸盐的葡甲胺盐,它是一种有机的、碘化的、不透射线的 X 射线造影剂,用于放射诊断。
T13198 Transcrocetin meglumine salt

trans-Crocetin meglumine salt

Others Others
Transcrocetin meglumine salt is a natural product isolated from saffron (Crocus sativus L.) and is a high-affinity antagonist of the NMDA receptor.
T32184 Iothalamate meglumine

Cysto-Conray,Methylglucamine iotalamate,EINECS 235-998-9,Meglumine conray

Iothalamate meglumine, known as radiopaque medium, can be used for urography, angiography, venography, and myelography. It is highly viscous and can bind to plasma proteins.
T32168 Iodamide Meglumine

Opacist E.R.,Meglumine iodamide,Iodamide 300,Renovue-65,Isteropac E.R.

Iodamide Meglumine is a bioactive chemical.
T33916 Pentagastrin meglumine

Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.
T4506 Gadopentetate dimeglumine

Meglumine gadopentetate,SH-L-451A,Gd-DTPA,Gadopentetic acid dimeglumine,钆喷酸葡胺,Gadopentetic acid dimeglumine salt

Others Others
Gadopentetate dimeglumine (Gd-DTPA) 可用于核磁共振成像 (MRI) 中,使血管、器官和其他非骨组织能够更清晰地被看到。
T74593 Taragarestrant meglumine

Taragarestrant meglumine (D-0502) 是一种口服有效、选择性的雌激素受体 (estrogen receptor) 降解剂,展现了对各种ER+乳腺癌细胞系及移植模型的强大活性。
T1790 Fosaprepitant dimeglumine

福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt

Neurokinin receptor GPCR/G Protein; Neuroscience
Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。
T32179 Ioglycamic acid

BE-419,Ioglycamide,BE419,BE 419

Iodoxylic acid, a mixture of meglumine and sodium salts, is used to visualize the biliary tract as a radiopaque diagnostic aid.

化合物

Meglumine
Cat.No: T0503
Synonym: Meglumin,Methylglucamin,葡甲胺,葡萄糖甲胺,Methylglucamine
Target: Others
Delafloxacin meglumine
Cat.No: T8173
Synonym: ABT492 meglumine,德拉沙星葡甲胺,WQ-3034 meglumine,RX-3341 meglumine
Target: Antibacterial, Antibiotic
Flunixin meglumine
Cat.No: T1209
Synonym: Banamine,Finadyne,Flunixin meglumin,氟尼辛葡甲胺
Target: COX
tafamidis meglumine
Cat.No: T7582
Synonym: Fx-1006A,他发米帝司甲葡胺
Target: Others
Diatrizoate meglumine
Cat.No: T20637
Synonym: Reno,Renografin,Renovist,泛影葡胺,Hypaque,Renocal,Sinografin
Target: Others
Transcrocetin meglumine salt
Cat.No: T13198
Synonym: trans-Crocetin meglumine salt
Target: Others
Iothalamate meglumine
Cat.No: T32184
Synonym: Cysto-Conray,Methylglucamine iotalamate,EINECS 235-998-9,Meglumine conray
Target:
Iodamide Meglumine
Cat.No: T32168
Synonym: Opacist E.R.,Meglumine iodamide,Iodamide 300,Renovue-65,Isteropac E.R.
Target:
Pentagastrin meglumine
Cat.No: T33916
Synonym:
Target:
Gadopentetate dimeglumine
Cat.No: T4506
Synonym: Meglumine gadopentetate,SH-L-451A,Gd-DTPA,Gadopentetic acid dimeglumine,钆喷酸葡胺,Gadopentetic acid dimeglumine salt
Target: Others
Taragarestrant meglumine
Cat.No: T74593
Synonym:
Target:
Fosaprepitant dimeglumine
Cat.No: T1790
Synonym: 福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
Ioglycamic acid
Cat.No: T32179
Synonym: BE-419,Ioglycamide,BE419,BE 419
Target:
Cat. No. Product Name Target Signaling Pathways
T75267 Crocetin meglumine

Crocetin (Transcrocetin) meglumine 从藏红花 (Crocus sativus L.) 中提取的,是一种高亲和力的 NMDA 受体拮抗剂。

天然产物

Crocetin meglumine
Cat.No: T75267
Synonym:
Target:
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