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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T76118 Malate dehydrogenase

Malate dehydrogenase 催化草酰乙酸盐和苹果酸盐的相互转化,与二核苷酸辅酶的氧化/还原相关。
T35520 Aflatoxin G1-13C17

Aflatoxin G1-13C17

Aflatoxin G1-13C17is intended for use as an internal standard for the quantification of aflatoxin G1by GC- or LC-MS. Aflatoxin G1is a mycotoxin that has been found inA. terricola.1In vivo, aflatoxin G1is lethal to ducklings (LD50= 1.18 mg/kg).2It induces hepatocellular carcinoma tumor formation and lethality in rats when administered at doses of 1.4 and 3 mg/animal, respectively. Aflatoxin G1also inhibits liver and kidney succinate dehydrogenase and fumarase, as well as kidney cytochrome oxidase...

化合物

Malate dehydrogenase
Cat.No: T76118
Synonym:
Target:
Aflatoxin G1-13C17
Cat.No: T35520
Synonym: Aflatoxin G1-13C17
Target:
Cat. No. Product Name Target Signaling Pathways
T8198 Visnagin

Others Others
Visnagin 是一种抗氧化剂呋喃香豆素衍生物。它具有预防Cerulein 诱导的急性胰腺炎的潜力。它在血管平滑肌中具有良好的血管扩张作用。它具有抗炎作用,可用于缓解疼痛的研究。
T4862 Oxaloacetic acid

Endogenous Metabolite Metabolism
Oxaloacetic acid 是一种代谢中间体,涉及多种途径,如葡萄糖异生、柠檬酸循环、乙醛酸循环、尿素循环、氨基酸合成和脂肪酸合成。
T15638 K-252c

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 μM). K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells.

天然产物

Visnagin
Cat.No: T8198
Synonym:
Target: Others
Oxaloacetic acid
Cat.No: T4862
Synonym:
Target: Endogenous Metabolite
K-252c
Cat.No: T15638
Synonym:
Target: PKC
TargetMol Loading
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