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Cat. No. Product Name Target Signaling Pathways
T39929 MS21

PROTACs PROTAC
MS21 is a unique AKT degrader that selectively hampers the proliferation of cancers with mutations in the PI3K/PTEN pathway, alongside wild-type KRAS and BRAF.
T5828 MS21570

5-(苄基硫代)-N-甲基-1,3,4-噻二唑-2-胺

GPR Endocrinology/Hormones; GPCR/G Protein
MS21570 作为 GPR171 拮抗剂基于其阻断能力,IC50 为 220 nM,可减少小鼠的焦虑样行为和恐惧条件反射。
T67746 IMS2186

Others Others
IMS2186 是一种抗脉络膜新生血管 (CNV) 试剂, 可以使癌细胞周期阻滞在 G2/M 期,由此产生抗增殖和抗血管生成作用。IMS2186 能够减少眼睛渗漏和病变细胞的数量,并且无眼内毒性。
T24501 MS2126

NSC 71584,NSC71584,MS 2126,MS-2126,NSC-71584

MS2126 is a Human p53 and CREB Binding Protein interaction inhibitor.
T28114 MS2177

MS 2177,MS-2177

MS2177 is a potent and selective inhibitor of SETD8, the only methyltransferase known to catalyze monomethylation of histone H4 lysine 20 (H4K20). MS2177 has an in vitro IC50 of 1.9 μM (σ = 1.05 μM, n = 4) in ascintillation proximity assay. Binding of MS2

化合物

MS21
Cat.No: T39929
Synonym:
Target: PROTACs
MS21570
Cat.No: T5828
Synonym: 5-(苄基硫代)-N-甲基-1,3,4-噻二唑-2-胺
Target: GPR
IMS2186
Cat.No: T67746
Synonym:
Target: Others
MS2126
Cat.No: T24501
Synonym: NSC 71584,NSC71584,MS 2126,MS-2126,NSC-71584
Target:
MS2177
Cat.No: T28114
Synonym: MS 2177,MS-2177
Target:
TargetMol Loading
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