Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0098 |
Quiflapon sodium
喹夫拉朋钠,MK591 |
FLAP | Immunology/Inflammation |
Quiflapon sodium (MK591) is a selective inhibitor of 5-Lipoxygenase-activating protein (FLAP). | |||
T16087 |
Quiflapon
喹夫拉朋,MK-591 |
Apoptosis; FLAP | Apoptosis; Immunology/Inflammation |
Quiflapon (MK-591) 是一种选择性和特异性的FLAP 抑制剂,可诱导细胞凋亡。它也是口服白三烯生物合成抑制剂,在完整的人和诱导的大鼠多形核白细胞 PMNLs 中,其IC50值分别为 3.1 nM 和 6.1 nM。 |