Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2509 |
Tozasertib
MK-0457,VX 680 |
Aurora Kinase; Autophagy | Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic |
Tozasertib (MK-0457) 是一种 Aurora A/B/C 激酶抑制剂,Ki 值分别为 0.6、18和4.6 nM。它显示出对 190 多种不同激酶的选择性。 | |||
T68415 |
Tozasertib lactate
|
||
Tozasertib lactate is a potent and selective small-molecule inhibitor of the Aurora kinases which suppresses tumor growth by inducing apoptosis in tumor cells in which Aurora kinases are overexpressed. |