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Cat. No. Product Name Target Signaling Pathways
T4628 Seladelpar

MBX 8025

PPAR DNA Damage/DNA Repair; Metabolism
Seladelpar (MBX 8025) 是一种有效的,具有口服活性的, 特异性PPAR-δ激动剂,EC50为 2 nM。
T35799 MBX-8025 (sodium salt)

MBX-8025 is an agonist of peroxisome proliferator-activated receptor δ (PPARδ).1 It is greater than 750- and 2,500-fold selective for PPARδ over PPARα and PPARγ. MBX-8025 (10 mg/kg per day for eight weeks) reduces increases in fasting blood glucose and serum insulin levels, and decreases insulin resistance in Alms1 mutant (foz/foz) mice fed an atherogenic diet as a model of diet-induced obesity, type 2 diabetes, and non-alcoholic steatohepatitis (NASH).2 It also decreases serum alanine transamin...
T68319 MBX-8025 lysine anhydrous

MBX-8025 lysine anhydrous is a selective PPAR-delta agonist.
T26182 Seladelpar lysine

MBX-8025 lysine dihydrate,MBX-8025 Lysine,MBX 8025 Lysine MBX8025 Lysine

Seladelpar lysine, a selective PPAR-δ agonist, is used for the therapy of Homozygous Familial Hypercholesterolemia (HoFH).
T12876 Seladelpar sodium salt

RWJ-800025 sodium salt,MBX-8025 sodium salt

Others Others
Seladelpar sodium salt (MBX-8025) 是一种具有口服活性、有效且特异性的PPARδ激动剂,EC50值为 2 nM。它对 PPARδ 的选择性分别是对 PPARα 和 PPARγ 的 750 和 2500 多倍。

化合物

Seladelpar
Cat.No: T4628
Synonym: MBX 8025
Target: PPAR
MBX-8025 (sodium salt)
Cat.No: T35799
Synonym:
Target:
MBX-8025 lysine anhydrous
Cat.No: T68319
Synonym:
Target:
Seladelpar lysine
Cat.No: T26182
Synonym: MBX-8025 lysine dihydrate,MBX-8025 Lysine,MBX 8025 Lysine MBX8025 Lysine
Target:
Seladelpar sodium salt
Cat.No: T12876
Synonym: RWJ-800025 sodium salt,MBX-8025 sodium salt
Target: Others
TargetMol Loading
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