Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15773 |
Lofepramine
Gamanil,洛非帕明,Amplit,Leo 640,Lopramine |
5-HT Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Lofepramine (Leo 640) 是一种有效的三环抗抑郁药,广泛地代谢为 Desipramine。它能够抑制摄取促进去甲肾上腺素能神经传递,以及抑制神经元摄取 5-羟色胺和色氨酸吡咯酶,增强 5-羟色胺能神经传递,进而发挥其抗抑郁作用。它还具有显著的抗焦虑效果。 | |||
T24414 |
Lofepramine hydrochloride
WHR-2908A,DB-2182,WHR 2908A |
||
Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative. |