Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6063 |
LY-411575
LY411575 |
Apoptosis; Gamma-secretase | Apoptosis; Neuroscience; Proteases/Proteasome; Stem Cells |
LY-411575 是一种高效的γ-secretase 抑制剂,能够抑制 Aβ40 蛋白的产生,在膜中的 IC50 为 0.078 nM,在细胞中为 0.082 nM。 它还抑制 Notch 切割,IC50 为 0.39 nM。 | |||
T11903 |
LY-411575 isomer 1
|
Others | Others |
LY-411575 isomer 1 is a potent γ-secretase inhibitor. LY-411575 isomer 1 is an isomer of LY411575. | |||
T11905 |
LY-411575 isomer 3
|
Others | Others |
LY-411575 isomer 3 is a potent γ-secretase inhibitor. LY-411575 isomer 3 is an isomer of LY411575. | |||
T11904 | LY-411575 isomer 2 | Others | Others |
LY-411575 isomer 2 is a potent γ-secretase inhibitor. LY-411575 isomer 2 is an isomer of LY411575. | |||
T63150 | LY-411575 (isomer 3) | ||
LY-411575 isomer 3 是 LY411575 的异构体。其中 LY411575 是一种高效的 γ-secretase 抑制剂。 | |||
T63149 | LY-411575 (isomer 2) | ||
LY-411575 isomer 2 是 LY411575 的异构体。其中 LY411575 是一种高效的 γ-secretase 抑制剂。 |