Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6022 |
LY404039
pomaglumetad |
Glucocorticoid Receptor; GluR | Endocrinology/Hormones; Neuroscience |
LY404039 (pomaglumetad) 是可口服的mGluR2和mGluR3选择性激动剂,有抗精神病和抗焦虑的作用。它对重组人mGluR2和mGluR3的Ki 分别为 149 和 92 nM,比对其他受体/转运蛋白的抑制性高 100 倍以上。 | |||
T61972 |
Pomaglumetad methionil hydrochloride
LY2140023 hydrochloride |
GluR | Neuroscience |
Pomaglumetad methionil hydrochloride (LY2140023 hydrochloride) (LY2140023 hydrochloride) 是的 LY404039 的蛋氨酸前药,具有口服活性。LY404039是一种选择性 mGlu2/3 受体激动剂。Pomaglumetad methionil hydrochloride 可用于精神分裂症的研究。 | |||
T11907 |
Pomaglumetad methionil anhydrous
LY2140023 |
GluR | Neuroscience |
LY2140023 has the potential for schizophrenia.LY2140023 is an orally active prodrug of LY404039. LY404039 is a selective metabotropic glutamate 2/3 receptor agonist. | |||
T12520 |
Pomaglumetad methionil
LY2140023 hydrate |
GluR | Neuroscience |
Pomaglumetad methionil is an oral methionine prodrug of the potent specific agonist of mGlu2/3 receptor LY404039. |