Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T27939 |
LY2940094 tartrate
LY2940094,LY 2940094,LY-2940094 tartrate,LY-2940094 |
||
LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism. | |||
T15799 |
LY2940094
LY-2940094 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
LY2940094 (LY-2940094) 是一种口服有效的选择性 NOP 受体拮抗剂,可降低动物模型的自身给药酒精依赖,对 NOP 受体具有高亲和力,Ki 为 0.105 nM,和拮抗活力,Kb 为 0.166 nM。 |