Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80116 |
LHRH
|
GNRH Receptor | GPCR/G Protein |
LHRH是一种调节生殖功能的下丘脑神经肽,常用于癌症研究。 | |||
T25105 |
APTAA-LHRH
Org-31276,Org31276,APTAALHRH,Org 31276 |
||
APTAA-LHRH is a gonadorelin antagonist. | |||
T25715 |
LHRH, Ala(6)-
L 1868,L-1868,L1868 |
||
LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent. | |||
T25808 |
MI 1544
Attcpl-LHRH,AttcplLHRH,MI-1544,MI1544,Attcpl LHRH |
||
MI 1544 is a LHRH antagonist. | |||
T25154 |
Bim 21009
LHRH-Ncpapa,Bim-21009,Bim21009,LHRHNcpapa,LHRH Ncpapa |
||
Bim 21009 is an inhibitor of gonadorelin. | |||
T26239 |
Surfagon
TAP 127,AY-25,205,LHRH-A2,AY 25,205,AY25,205 |
||
Surfagon is an effective LHRH agonist. | |||
T76617 |
(D-Trp6)-LHRH free acid
|
||
(D-Trp6)-LHRH free acid 是促黄体生成素释放激素 (LHRH) 激动剂。 | |||
T76616 |
(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
|
||
(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH 是一种黄体生成素释放激素 (LHRH) 的类似物,主要通过促进垂体分泌黄体生成素 (LH) 和促卵泡激素 (FSH) 来在生殖调控中发挥关键作用。 | |||
T76593 |
(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)
|
||
'(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)' 为一种GnRH类似物,主要用于诱导养殖鱼类排卵和/或产卵。 | |||
T76620 |
(D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH
|
||
(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH 是黄体生成素释放激素 (LHRH) 的类似物。LHRH 通过刺激垂体黄体生成素 (LH) 和促卵泡激素 (FSH) 的释放,在控制生殖中发挥核心作用。 | |||
T76615 |
(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH
|
||
(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH是一种LHRH(黄体生成素释放激素)的类似物,主要通过激活垂体分泌黄体生成素(LH)和促卵泡激素(FSH)来在生殖调控中发挥核心作用。 | |||
TP1112L |
LH-RH, salmon acetate(86073-88-3 free base)
Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate |
Others | Others |
LH-RH, salmon acetate(86073-88-3 free base) (Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate) 是一种在下丘脑中合成的垂体激素,在控制生殖功能中起着至关重要的作用。 | |||
TP1648L |
[Gln8]-C517 (LH-RH), chicken acetate
[Gln8]-C517 (LH-RH), chicken acetate(47922-48-5 free base) |
Others | Others |
[Gln8]-C517 (LH-RH), chicken acetate(47922-48-5 free base) 是一种鸟类下丘脑肽,可刺激垂体前叶释放促性腺激素,从而调节生殖功能。 | |||
TP1648 |
[Gln8]-C517 (LH-RH), chicken
|
||
[Gln8] Luteinizing hormone releasing hormone ([Gln8] LH-RH), Avian hypothalamic peptide that stimulates release of gonadotropins from anterior pituitary, thus regulating reproductive functions. | |||
TP1112 |
Luteinizing Hormone Releasing Hormone (LH-RH), salmon
LH-RH, salmon |
||
Luteinizing Hormone Releasing Hormone (LH-RH) is a pituitary Hormone synthesized in the hypothalamus and plays a crucial role in the control of reproductive function. | |||
T3538 |
Sufugolix
TAK-013 |
LHRH | Endocrinology/Hormones |
Sufugolix (TAK-013) 是一种高效的、有口服活性的黄体激素释放激素(LHRH) 受体拮抗剂(IC50:0.1 nM)。 | |||
T9380L |
Antide acetate
安替肽,Antide acetate (112568-12-4 Free base) |
LHRH | Endocrinology/Hormones |
Antide acetate 是一种 LHRH 拮抗剂,可抑制垂体释放 LH 和 FSH。 | |||
T4102 |
Goserelin acetate
醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex |
Apoptosis; GNRH Receptor | Apoptosis; GPCR/G Protein |
Goserelin acetate (Fertilan) 是一种促性腺激素释放激素 (GnRH/LHRH) 十肽类似物,能作为GnRH 激动剂。它可研究乳腺癌、上皮性卵巢癌和前列腺癌。 | |||
T3630 |
Relugolix
RVT-601,瑞卢戈利,TAK-385 |
GNRH Receptor | GPCR/G Protein |
Relugolix (RVT-601) 是口服有活性的非肽性促性腺激素释放激素的拮抗剂。同 TAK-013 相比,它对人和猴子的受体具有高亲和力和强拮抗活性,它们的 IC50值分别为0.33 nM 和0.32 nM。它可用于研究性激素依赖性疾病,如子宫肌瘤、子宫内膜异位症、前列腺癌等。 | |||
T26040 |
Ramorelix
HOE 013,HOE013,HOE-013 |
||
Ramorelix is an antagonist of luteinizing hormone-releasing hormone (LHRH). | |||
T68420 |
Detirelix
|
||
Detirelix is an LHRH antagonist. | |||
T26444 |
A 76154
A-76154,A76154 |
||
A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH). | |||
T28954 |
Teverelix
|
||
Teverelix is a water-soluble antagonist of luteinizing hormone-releasing hormone (LHRH). | |||
T76350 |
[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
|
||
[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH 是一种黄体激素释放激素 (LHRH) 类似物,可作为 GnRH 受体拮抗剂。 | |||
T26135 |
RS 18286
RS18286,RS-18286 |
||
RS 18286 is a LHRH antagonist. | |||
T71592 | Detirelix acetate | ||
Detirelix acetate is an LHRH Antagonist | |||
T23412 |
T 98475
|
Others | Others |
gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active | |||
T70819 | Argtide | ||
Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist. | |||
T76354 |
LH-RH (4-10)
|
||
LH-RH (4-10),一种性腺激素释放激素(LHRH)的主要降解产物,属于七肽类,主要在巨噬细胞和II型肺细胞中产生。 | |||
T76349 |
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
|
||
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide 是 LHRH 多肽类似物。 | |||
T76322 |
LH-RH II (chicken)
|
||
LH-RH II (chicken) 为家鸡下丘脑黄体生成素释放激素(LHRH)两种形式之一,亦为哺乳动物LHRH的结构变体。该化合物促进家鸡促性腺激素释放。 | |||
T76558 |
Onvitrelin ucalontide
|
||
Onvitrelin ucalontide ([Phor18-LHRH (338613)]) 是一种 LHRH (黄体生成素释放激素) 的类似物,展现出抗肿瘤特性。这一化合物是一个具备序列 KFAKFAKKFAKFAKKFAKQHWSYGLRPG 的肽,能在小鼠模型上有效地抑制乳腺癌、卵巢癌和前列腺癌的异种移植物生长。 | |||
T76348 |
[D-Lys6]-LH-RH
|
||
[D-Lys6]-LH-RH 是一种黄体激素释放激素 (LHRH) 类似物,可作为GnRH 受体激动剂。 | |||
T76353 |
LH-RH (7-10)
|
||
LH-RH (7-10),一种由性腺激素释放激素 (LHRH) 在垂体和下丘脑降解过程中形成的主要四肽降解产物之一,存在于巨噬细胞、I 型样及II 型肺细胞中。 | |||
T83499 |
[D-Phe2,6, Pro3]-LH-RH
|
||
[D-Phe2,6, Pro3]-LH-RH是一种促黄体生成素释放激素(LHRH)的高效拮抗剂,具有特定氨基酸序列变异。 | |||
T76351 | [D-Ala6]-LH-RH | ||
[D-Ala6]-LH-RH,一种黄体激素释放激素(LHRH)模拟物,充当GnRH受体的激动剂。 | |||
T69492 |
Ozarelix
|
||
Ozarelix is a fourth generation GnRH antagonist, induces apoptosis in hormone refractory androgen receptor negative prostate cancer cells modulating expression and activity of death receptors. Mechanistically, LHRH antagonists exert rapid inhibition of luteinizing hormone and follicle stimulating hormone with an accompanying rapid decrease in sex hormones and would therefore be expected to be effective in a variety of hormonally dependent disease states including ovarian cancer, prostate cancer,... | |||
TP1342 |
GnRH-I
|
||
GnRH-I is a small 10 amino acid long peptide (decapeptide) from the hypothalamus,It is also known as luteinizing hormone releasing hormone (LHRH), is a key molecule in the regulation of reproduction in vertebrates. GnRH, a decapeptide, is produced by neur | |||
T70775 |
Zoptarelin doxorubicin
|
||
Zoptarelin doxorubicin, also known as AEZS-108, is an LHRH agonist. Zoptarelin doxorubicin is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R) that is conjugated to the anthracycline antibiotic doxorubicin with potential antineoplastic activity. Zoptarelin doxorubicin binds to GnRH-1Rs, which may be highly expressed on endometrial and ovarian tumor cell membrane surfaces, and is internalized. Once inside the cell, the doxorubicin moiety of this agent intercalates in... |