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Cat. No. Product Name Target Signaling Pathways
T80116 LHRH

GNRH Receptor GPCR/G Protein
LHRH是一种调节生殖功能的下丘脑神经肽,常用于癌症研究。
T25105 APTAA-LHRH

Org-31276,Org31276,APTAALHRH,Org 31276

APTAA-LHRH is a gonadorelin antagonist.
T25715 LHRH, Ala(6)-

L 1868,L-1868,L1868

LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.
T25808 MI 1544

Attcpl-LHRH,AttcplLHRH,MI-1544,MI1544,Attcpl LHRH

MI 1544 is a LHRH antagonist.
T25154 Bim 21009

LHRH-Ncpapa,Bim-21009,Bim21009,LHRHNcpapa,LHRH Ncpapa

Bim 21009 is an inhibitor of gonadorelin.
T26239 Surfagon

TAP 127,AY-25,205,LHRH-A2,AY 25,205,AY25,205

Surfagon is an effective LHRH agonist.
T76617 (D-Trp6)-LHRH free acid

(D-Trp6)-LHRH free acid 是促黄体生成素释放激素 (LHRH) 激动剂。
T76616 (D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH

(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH 是一种黄体生成素释放激素 (LHRH) 的类似物,主要通过促进垂体分泌黄体生成素 (LH) 和促卵泡激素 (FSH) 来在生殖调控中发挥关键作用。
T76593 (Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)

'(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)' 为一种GnRH类似物,主要用于诱导养殖鱼类排卵和/或产卵。
T76620 (D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH

(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH 是黄体生成素释放激素 (LHRH) 的类似物。LHRH 通过刺激垂体黄体生成素 (LH) 和促卵泡激素 (FSH) 的释放,在控制生殖中发挥核心作用。
T76615 (D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH

(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH是一种LHRH(黄体生成素释放激素)的类似物,主要通过激活垂体分泌黄体生成素(LH)和促卵泡激素(FSH)来在生殖调控中发挥核心作用。
TP1112L LH-RH, salmon acetate(86073-88-3 free base)

Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate

Others Others
LH-RH, salmon acetate(86073-88-3 free base) (Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate) 是一种在下丘脑中合成的垂体激素,在控制生殖功能中起着至关重要的作用。
TP1648L [Gln8]-C517 (LH-RH), chicken acetate

[Gln8]-C517 (LH-RH), chicken acetate(47922-48-5 free base)

Others Others
[Gln8]-C517 (LH-RH), chicken acetate(47922-48-5 free base) 是一种鸟类下丘脑肽,可刺激垂体前叶释放促性腺激素,从而调节生殖功能。
TP1648 [Gln8]-C517 (LH-RH), chicken

[Gln8] Luteinizing hormone releasing hormone ([Gln8] LH-RH), Avian hypothalamic peptide that stimulates release of gonadotropins from anterior pituitary, thus regulating reproductive functions.
TP1112 Luteinizing Hormone Releasing Hormone (LH-RH), salmon

LH-RH, salmon

Luteinizing Hormone Releasing Hormone (LH-RH) is a pituitary Hormone synthesized in the hypothalamus and plays a crucial role in the control of reproductive function.
T3538 Sufugolix

TAK-013

LHRH Endocrinology/Hormones
Sufugolix (TAK-013) 是一种高效的、有口服活性的黄体激素释放激素(LHRH) 受体拮抗剂(IC50:0.1 nM)。
T9380L Antide acetate

安替肽,Antide acetate (112568-12-4 Free base)

LHRH Endocrinology/Hormones
Antide acetate 是一种 LHRH 拮抗剂,可抑制垂体释放 LH 和 FSH。
T4102 Goserelin acetate

醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex

Apoptosis; GNRH Receptor Apoptosis; GPCR/G Protein
Goserelin acetate (Fertilan) 是一种促性腺激素释放激素 (GnRH/LHRH) 十肽类似物,能作为GnRH 激动剂。它可研究乳腺癌、上皮性卵巢癌和前列腺癌。
T3630 Relugolix

RVT-601,瑞卢戈利,TAK-385

GNRH Receptor GPCR/G Protein
Relugolix (RVT-601) 是口服有活性的非肽性促性腺激素释放激素的拮抗剂。同 TAK-013 相比,它对人和猴子的受体具有高亲和力和强拮抗活性,它们的 IC50值分别为0.33 nM 和0.32 nM。它可用于研究性激素依赖性疾病,如子宫肌瘤、子宫内膜异位症、前列腺癌等。
T26040 Ramorelix

HOE 013,HOE013,HOE-013

Ramorelix is an antagonist of luteinizing hormone-releasing hormone (LHRH).
T68420 Detirelix

Detirelix is an LHRH antagonist.
T26444 A 76154

A-76154,A76154

A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).
T28954 Teverelix

Teverelix is a water-soluble antagonist of luteinizing hormone-releasing hormone (LHRH).
T76350 [D-Glp1,D-Phe2,D-Trp3,6]-LH-RH

[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH 是一种黄体激素释放激素 (LHRH) 类似物,可作为 GnRH 受体拮抗剂。
T26135 RS 18286

RS18286,RS-18286

RS 18286 is a LHRH antagonist.
T71592 Detirelix acetate

Detirelix acetate is an LHRH Antagonist
T23412 T 98475

Others Others
gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active
T70819 Argtide

Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.
T76354 LH-RH (4-10)

LH-RH (4-10),一种性腺激素释放激素(LHRH)的主要降解产物,属于七肽类,主要在巨噬细胞和II型肺细胞中产生。
T76349 [D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide

[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide 是 LHRH 多肽类似物。
T76322 LH-RH II (chicken)

LH-RH II (chicken) 为家鸡下丘脑黄体生成素释放激素(LHRH)两种形式之一,亦为哺乳动物LHRH的结构变体。该化合物促进家鸡促性腺激素释放。
T76558 Onvitrelin ucalontide

Onvitrelin ucalontide ([Phor18-LHRH (338613)]) 是一种 LHRH (黄体生成素释放激素) 的类似物,展现出抗肿瘤特性。这一化合物是一个具备序列 KFAKFAKKFAKFAKKFAKQHWSYGLRPG 的肽,能在小鼠模型上有效地抑制乳腺癌、卵巢癌和前列腺癌的异种移植物生长。
T76348 [D-Lys6]-LH-RH

[D-Lys6]-LH-RH 是一种黄体激素释放激素 (LHRH) 类似物,可作为GnRH 受体激动剂。
T76353 LH-RH (7-10)

LH-RH (7-10),一种由性腺激素释放激素 (LHRH) 在垂体和下丘脑降解过程中形成的主要四肽降解产物之一,存在于巨噬细胞、I 型样及II 型肺细胞中。
T83499 [D-Phe2,6, Pro3]-LH-RH

[D-Phe2,6, Pro3]-LH-RH是一种促黄体生成素释放激素(LHRH)的高效拮抗剂,具有特定氨基酸序列变异。
T76351 [D-Ala6]-LH-RH

[D-Ala6]-LH-RH,一种黄体激素释放激素(LHRH)模拟物,充当GnRH受体的激动剂。
T69492 Ozarelix

Ozarelix is a fourth generation GnRH antagonist, induces apoptosis in hormone refractory androgen receptor negative prostate cancer cells modulating expression and activity of death receptors. Mechanistically, LHRH antagonists exert rapid inhibition of luteinizing hormone and follicle stimulating hormone with an accompanying rapid decrease in sex hormones and would therefore be expected to be effective in a variety of hormonally dependent disease states including ovarian cancer, prostate cancer,...
TP1342 GnRH-I

GnRH-I is a small 10 amino acid long peptide (decapeptide) from the hypothalamus,It is also known as luteinizing hormone releasing hormone (LHRH), is a key molecule in the regulation of reproduction in vertebrates. GnRH, a decapeptide, is produced by neur
T70775 Zoptarelin doxorubicin

Zoptarelin doxorubicin, also known as AEZS-108, is an LHRH agonist. Zoptarelin doxorubicin is a peptide agonist of the gonadotropin releasing hormone-1 receptor (GnRH-1R) that is conjugated to the anthracycline antibiotic doxorubicin with potential antineoplastic activity. Zoptarelin doxorubicin binds to GnRH-1Rs, which may be highly expressed on endometrial and ovarian tumor cell membrane surfaces, and is internalized. Once inside the cell, the doxorubicin moiety of this agent intercalates in...

化合物

LHRH
Cat.No: T80116
Synonym:
Target: GNRH Receptor
APTAA-LHRH
Cat.No: T25105
Synonym: Org-31276,Org31276,APTAALHRH,Org 31276
Target:
LHRH, Ala(6)-
Cat.No: T25715
Synonym: L 1868,L-1868,L1868
Target:
MI 1544
Cat.No: T25808
Synonym: Attcpl-LHRH,AttcplLHRH,MI-1544,MI1544,Attcpl LHRH
Target:
Bim 21009
Cat.No: T25154
Synonym: LHRH-Ncpapa,Bim-21009,Bim21009,LHRHNcpapa,LHRH Ncpapa
Target:
Surfagon
Cat.No: T26239
Synonym: TAP 127,AY-25,205,LHRH-A2,AY 25,205,AY25,205
Target:
(D-Trp6)-LHRH free acid
Cat.No: T76617
Synonym:
Target:
(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
Cat.No: T76616
Synonym:
Target:
(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)
Cat.No: T76593
Synonym:
Target:
(D-Tyr5,D-Ser(tBu)6,Azagly10)-LHRH
Cat.No: T76620
Synonym:
Target:
(D-Ser(tBu)6,D-Leu7,Azagly10)-LHRH
Cat.No: T76615
Synonym:
Target:
LH-RH, salmon acetate(86073-88-3 free base)
Cat.No: TP1112L
Synonym: Luteinizing Hormone Releasing Hormone (LH-RH), salmon acetate
Target: Others
[Gln8]-C517 (LH-RH), chicken acetate
Cat.No: TP1648L
Synonym: [Gln8]-C517 (LH-RH), chicken acetate(47922-48-5 free base)
Target: Others
[Gln8]-C517 (LH-RH), chicken
Cat.No: TP1648
Synonym:
Target:
Luteinizing Hormone Releasing Hormone (LH-RH), salmon
Cat.No: TP1112
Synonym: LH-RH, salmon
Target:
Sufugolix
Cat.No: T3538
Synonym: TAK-013
Target: LHRH
Antide acetate
Cat.No: T9380L
Synonym: 安替肽,Antide acetate (112568-12-4 Free base)
Target: LHRH
Goserelin acetate
Cat.No: T4102
Synonym: 醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex
Target: Apoptosis, GNRH Receptor
Relugolix
Cat.No: T3630
Synonym: RVT-601,瑞卢戈利,TAK-385
Target: GNRH Receptor
Ramorelix
Cat.No: T26040
Synonym: HOE 013,HOE013,HOE-013
Target:
Detirelix
Cat.No: T68420
Synonym:
Target:
A 76154
Cat.No: T26444
Synonym: A-76154,A76154
Target:
Teverelix
Cat.No: T28954
Synonym:
Target:
[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
Cat.No: T76350
Synonym:
Target:
RS 18286
Cat.No: T26135
Synonym: RS18286,RS-18286
Target:
Detirelix acetate
Cat.No: T71592
Synonym:
Target:
T 98475
Cat.No: T23412
Synonym:
Target: Others
Argtide
Cat.No: T70819
Synonym:
Target:
LH-RH (4-10)
Cat.No: T76354
Synonym:
Target:
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
Cat.No: T76349
Synonym:
Target:
LH-RH II (chicken)
Cat.No: T76322
Synonym:
Target:
Onvitrelin ucalontide
Cat.No: T76558
Synonym:
Target:
[D-Lys6]-LH-RH
Cat.No: T76348
Synonym:
Target:
LH-RH (7-10)
Cat.No: T76353
Synonym:
Target:
[D-Phe2,6, Pro3]-LH-RH
Cat.No: T83499
Synonym:
Target:
[D-Ala6]-LH-RH
Cat.No: T76351
Synonym:
Target:
Ozarelix
Cat.No: T69492
Synonym:
Target:
GnRH-I
Cat.No: TP1342
Synonym:
Target:
Zoptarelin doxorubicin
Cat.No: T70775
Synonym:
Target:
TargetMol Loading
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