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4

抑制剂 & 化合物

4

天然产物

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Cat. No. Product Name Target Signaling Pathways
T12368 Pasireotide L-aspartate salt

帕瑞肽天门冬氨酸盐,SOM230 L-aspartate

Others Others
Pasireotide L-aspartate salt is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively).
T12370 Pasireotide

SOM 230,SOM 320,帕瑞肽

Others Others
Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively).
T28298 Pasireotide diaspartate

SOM-230,SOM230,trade name: Signifor,SOM 230,Signifor LAR

Pasireotide is a somatostatin analog with a 40-fold increased affinity to somatostatin receptor 5 compared to other somatostatin analogs.
T13811 Pasireotide ditrifluoroacetate

SOM230 ditrifluoroacetate,Pasireotide ditrifluoroacetate (396091-73-9 free base),Pasireotide TFA salt

Others Others
Pasireotide is a stable cyclohexapeptide somatostatin mimic.

化合物

Pasireotide L-aspartate salt
Cat.No: T12368
Synonym: 帕瑞肽天门冬氨酸盐,SOM230 L-aspartate
Target: Others
Pasireotide
Cat.No: T12370
Synonym: SOM 230,SOM 320,帕瑞肽
Target: Others
Pasireotide diaspartate
Cat.No: T28298
Synonym: SOM-230,SOM230,trade name: Signifor,SOM 230,Signifor LAR
Target:
Pasireotide ditrifluoroacetate
Cat.No: T13811
Synonym: SOM230 ditrifluoroacetate,Pasireotide ditrifluoroacetate (396091-73-9 free base),Pasireotide TFA salt
Target: Others
Cat. No. Product Name Target Signaling Pathways
T5287 N-Acetyl-L-aspartic acid

AC-ASP-OH,N-Acetylaspartic acid,N-乙酰-L-天门冬氨酸

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-aspartic acid (AC-ASP-OH) 是天冬氨酸的衍生物, 是由氨基酸天冬氨酸和乙酰辅酶 A 在神经元中合成的。
T2O2774 L-Asparagine

alpha-aminosuccinamic acid,L-天门冬氨酸,(-)-Asparagine,Asparamide,2-Aminosuccinamic acid,Asn,Altheine

Endogenous Metabolite Metabolism
L-Asparagine (Asparamide) 是一种非必需氨基酸,可以参与神经和脑组织细胞功能的代谢控制。
T4885 (-)-Aspartic acid

(R)-Aspartic acid,Asp,D-(-)-Aspartic acid,D-天门冬氨酸,Aminosuccinic acid,asparagic acid,L-Homoproline,D-Aspartic acid

Endogenous Metabolite; NMDAR; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
(-)-Aspartic acid (L-Homoproline) 是一种存在于无脊椎动物和脊椎动物中的内源性氨基酸,是 NMDA 受体激动剂,可调节睾酮合成。
T19554 L-Aspartic aicd sodium

L-Aspartic acid sodium,Sodium L-aspartate

Others; Sodium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
L-Aspartic aicd sodium (Sodium L-aspartate) 是一种氨基酸,是一种结肠特异性活性分子输送的前体活性分子,可促进大鼠前脑膜囊泡的 Na+外排。

天然产物

N-Acetyl-L-aspartic acid
Cat.No: T5287
Synonym: AC-ASP-OH,N-Acetylaspartic acid,N-乙酰-L-天门冬氨酸
Target: Others, Endogenous Metabolite
L-Asparagine
Cat.No: T2O2774
Synonym: alpha-aminosuccinamic acid,L-天门冬氨酸,(-)-Asparagine,Asparamide,2-Aminosuccinamic acid,Asn,Altheine
Target: Endogenous Metabolite
(-)-Aspartic acid
Cat.No: T4885
Synonym: (R)-Aspartic acid,Asp,D-(-)-Aspartic acid,D-天门冬氨酸,Aminosuccinic acid,asparagic acid,L-Homoproline,D-Aspartic acid
Target: Endogenous Metabolite, NMDAR, iGluR
L-Aspartic aicd sodium
Cat.No: T19554
Synonym: L-Aspartic acid sodium,Sodium L-aspartate
Target: Others, Sodium Channel, Endogenous Metabolite
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