Cat. No. | Product Name | Target | Signaling Pathways |
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T62784 |
KRAS inhibitor-18
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KRAS inhibitor-18 (compound 3-10) 是一种 KRAS G12C 的有效抑制剂 (IC50: 4.74 μM)。KRAS inhibitor-18 在 MIA PaCA-2,A549 细胞中表现出 p-ERK 抑制作用,IC50s 分别为 66.4,11.1 μM。KRAS inhibitor-18 具有潜力进行胰腺癌、结直肠癌和肺癌的研究。 | |||
T78212 |
RMC-9805
KRAS G12D inhibitor 18,KRAS G12D IN 18 |
Others | Others |
RMC-9805为一种有效的 KRAS G12D 抑制剂,具有潜在的抗肿瘤和抑制肿瘤细胞增殖的活性,可用于研究胰腺癌。 | |||
T40285 |
KRAS G12C inhibitor 18
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KRAS G12C inhibitor 18 is a potent, orally active compound that inhibits KRAS G12C and exhibits anti-tumor activities. | |||
T11768 |
KRAS G12C inhibitor 14
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Ras | GPCR/G Protein; MAPK |
KRAS G12C inhibitor 14 是一种有效的 KRAS G12C 抑制剂(IC50= 18 nM)。 |