Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11775 |
KRAS inhibitor-8
|
Ras | GPCR/G Protein; MAPK |
KRAS inhibitor-8 is a potent KRAS G12C inhibitor. | |||
T9585 |
GNE-9815
3-(2-cyanopropan-2-yl)-N-[2-fluoro-4-methyl-5-(7-methyl-8-oxo-7,8-dihydropyrido[2,3-d]pyridazin-3-yl)phenyl]benzamide |
Raf | MAPK |
GNE-9815 (3-(2-cyanopropan-2-yl)-N-[2-fluoro-4-methyl-5-(7-methyl-8-oxo-7,8-dihydropyrido[2,3-d]pyridazin-3-yl)phenyl]benzamide) 是一种高激酶选择性 RAF 抑制剂,可用于通过联合治疗靶向 KRAS 突变癌症。 | |||
T74663 |
KRAS G12D inhibitor 17
|
||
KRAS G12D inhibitor 17 (example 8) 是一种喹唑啉连接 (4R)-4-羟基-l -脯氨酸酰胺化合物,可诱导 G12D 突变 KRAS 蛋白降解。KRAS G12D inhibitor 17 是一种 PTOTAC。 |