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Cat. No. Product Name Target Signaling Pathways
T11751 KDOAM-25

Antibacterial Microbiology/Virology
KDOAM-25, a potent and highly selective inhibitor of histone lysine demethylases 5 (KDM5) with IC50 values of 71 nM for KDM5A, 19 nM for KDM5B, 69 nM for KDM5C, and 69 nM for KDM5D, enhances global H3K4 methylation at transcriptional start sites and reduces proliferation in multiple myeloma MM1S cells.
T11750 KDOAM-25 citrate

Others Others
KDOAM-25 citrate 是有效且具有高选择性的组蛋白赖氨酸脱甲基酶 5 (KDM5) 抑制剂,对 KDM5A,KDM5B,KDM5C,KDM5D 的IC50分别为 71 nM,19 nM,69 nM,69 nM。用KDOAM-25 citrate 处理的多发性骨髓瘤 MM1S 细胞显示转录起始位点的整体 H3K4 甲基化增加,增殖受损。
T11750L KDOAM-25 trihydrochloride (2230731-99-2 free base)

KDOAM-25 trihydrochloride

Others Others
KDOAM-25 trihydrochloride increases global H3K4 methylation at transcriptional start sites and impairs proliferation in multiple myeloma MM1S cells. KDOAM-25 trihydrochloride is a potent and highly selective histone lysine demethylases 5 (KDM5) inhibitor
T62166 KDOAM-25 trihydrochloride

KDOAM-25 trihydrochloride 是一种有效的、高度选择性的组蛋白赖氨酸脱甲基酶 5 (KDM5) 抑制剂,能够作用于 KDM5A (IC50: 71 nM)、KDM5B (IC50: 19 nM)、KDM5C (IC50: 69 nM)、KDM5D (IC50: 69 nM)。KDOAM-25 trihydrochloride 能够提高转录起始位点的整体 H3K4 甲基化,可阻碍多发性骨髓瘤 MM1S 细胞的增殖。

化合物

KDOAM-25
Cat.No: T11751
Synonym:
Target: Antibacterial
KDOAM-25 citrate
Cat.No: T11750
Synonym:
Target: Others
KDOAM-25 trihydrochloride (2230731-99-2 free base)
Cat.No: T11750L
Synonym: KDOAM-25 trihydrochloride
Target: Others
KDOAM-25 trihydrochloride
Cat.No: T62166
Synonym:
Target:
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