Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T62166 | KDOAM-25 trihydrochloride | ||
KDOAM-25 trihydrochloride 是一种有效的、高度选择性的组蛋白赖氨酸脱甲基酶 5 (KDM5) 抑制剂,能够作用于 KDM5A (IC50: 71 nM)、KDM5B (IC50: 19 nM)、KDM5C (IC50: 69 nM)、KDM5D (IC50: 69 nM)。KDOAM-25 trihydrochloride 能够提高转录起始位点的整体 H3K4 甲基化,可阻碍多发性骨髓瘤 MM1S 细胞的增殖。 | |||
T11750L |
KDOAM-25 trihydrochloride (2230731-99-2 free base)
KDOAM-25 trihydrochloride |
Others | Others |
KDOAM-25 trihydrochloride increases global H3K4 methylation at transcriptional start sites and impairs proliferation in multiple myeloma MM1S cells. KDOAM-25 trihydrochloride is a potent and highly selective histone lysine demethylases 5 (KDM5) inhibitor |