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Cat. No. Product Name Target Signaling Pathways
T5484 GSK467

Histone Demethylase; Histone Methyltransferase Chromatin/Epigenetic
GSK467 是一种有效的、选择性的 KDM5 (JARID1) 抑制剂,Ki 值为10 nM。
T16435 PBIT

Histone Demethylase; Histone Methyltransferase Chromatin/Epigenetic
PBIT 是一种特异性 Jumonji/AT 富集互作结构域 1 抑制剂,抑制JARID1A 和JARID1C,IC50分别为 6 和 4.9 μM。它抑制JARID1B(KDM5B 或PLU1) 组蛋白去甲基化酶,IC50值约为 3 μM。
T61565 KDM5B-IN-3

KDM5B-IN-3 (Compound 5) is an inhibitor of histone lysine-specific demethylase 5B (KDM5B) or JARID1B. It effectively inhibits the activity of KDM5B with an IC50 value of 9.32 μM. Consequently, KDM5B-IN-3 serves as a valuable tool in gastric cancer research [1].

化合物

GSK467
Cat.No: T5484
Synonym:
Target: Histone Demethylase, Histone Methyltransferase
PBIT
Cat.No: T16435
Synonym:
Target: Histone Demethylase, Histone Methyltransferase
KDM5B-IN-3
Cat.No: T61565
Synonym:
Target:
TargetMol Loading
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