Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5484 |
GSK467
|
Histone Demethylase; Histone Methyltransferase | Chromatin/Epigenetic |
GSK467 是一种有效的、选择性的 KDM5 (JARID1) 抑制剂,Ki 值为10 nM。 | |||
T16435 |
PBIT
|
Histone Demethylase; Histone Methyltransferase | Chromatin/Epigenetic |
PBIT 是一种特异性 Jumonji/AT 富集互作结构域 1 抑制剂,抑制JARID1A 和JARID1C,IC50分别为 6 和 4.9 μM。它抑制JARID1B(KDM5B 或PLU1) 组蛋白去甲基化酶,IC50值约为 3 μM。 | |||
T61565 | KDM5B-IN-3 | ||
KDM5B-IN-3 (Compound 5) is an inhibitor of histone lysine-specific demethylase 5B (KDM5B) or JARID1B. It effectively inhibits the activity of KDM5B with an IC50 value of 9.32 μM. Consequently, KDM5B-IN-3 serves as a valuable tool in gastric cancer research [1]. |