Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T82017 |
JAK-IN-34
|
JAK | Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells |
JAK-IN-34 对JAKs具有有效抑制作用,其IC50值分别针对JAK1、JAK2、JAK3、TYK2为0.40、0.83、2.10、1.95 nM 。此外,JAK-IN-34 能够降低关节肿胀,并展现出良好的安全性。 | |||
T11704 |
JAK-IN-3
|
CCR | Immunology/Inflammation; Microbiology/Virology |
JAK-IN-3 is a potent JAK inhibitor, with IC50 values of 3 nM, 5 nM, 34 nM and 70 nM for JAK3, JAK1, TYK2 and JAK2, respectively. |