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Cat. No. Product Name Target Signaling Pathways
T1906 Molibresib

GSK 525762A,GSK525762,(4S)-6-(4-氯苯基)-N-乙基-8-甲氧基-1-甲基-4H-[1,2,4]三唑并[4,3-a][1,4]苯并二氮杂卓-4-乙酰胺,I-BET 762

Epigenetic Reader Domain Chromatin/Epigenetic
Molibresib (GSK525762) 是一种 BET 溴结构域抑制剂,IC50为32.5在42.5 nM 之间。
T11472L Molibresib besylate

I-BET 762 besylate,GSK 525762C

CCR Immunology/Inflammation; Microbiology/Virology
Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM).
T13086 I-BET762 carboxylic acid

Molibresib carboxylic acid,PROTAC BRD4-binding moiety 2,GSK525762A carboxylic acid

Epigenetic Reader Domain Chromatin/Epigenetic
I-BET762 carboxylic acid is an inhibitor of BRD4(pIC50 of 5.1).

化合物

Molibresib
Cat.No: T1906
Synonym: GSK 525762A,GSK525762,(4S)-6-(4-氯苯基)-N-乙基-8-甲氧基-1-甲基-4H-[1,2,4]三唑并[4,3-a][1,4]苯并二氮杂卓-4-乙酰胺,I-BET 762
Target: Epigenetic Reader Domain
Molibresib besylate
Cat.No: T11472L
Synonym: I-BET 762 besylate,GSK 525762C
Target: CCR
I-BET762 carboxylic acid
Cat.No: T13086
Synonym: Molibresib carboxylic acid,PROTAC BRD4-binding moiety 2,GSK525762A carboxylic acid
Target: Epigenetic Reader Domain
TargetMol Loading
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