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Cat. No. Product Name Target Signaling Pathways
T27527 HBF-0259

HBF 0259

Antiviral Immunology/Inflammation
HBF-0259 是有效的乙型肝炎病毒 表面抗原分泌选择性抑制剂,在 HepG2.2.15 细胞中的 EC50为 1.5 μM。
T60898 HbF inducer-1

HbF inducer-1 是一种胎儿血红蛋白诱导剂,具有口服生物活性。
T21652 RN-1 dihydrochloride

Histone Demethylase; MAO Chromatin/Epigenetic; Metabolism; Neuroscience
RN-1 dihydrochloride 是血脑屏障通透性的、不可逆的赖氨酸特异性脱甲基酶 1 (LSD1) 选择性抑制剂,IC50为 70 nM,对 LSD1 的选择性高于 MAO-A 和 MAO-B,IC50分别为 0.51 μM 和 2.785 μM。
T19583 TN1

Others Others
TN1 是一种有效的胎儿型血红蛋白 (HbF) 诱导剂。
T40154 FTX-6058

FTX-6058 is a potent orally active inhibitor targeting Embryonic Ectoderm Development (EED). It effectively induces HbF protein expression in both cell and murine models. This compound holds significant potential for researching select hemoglobinopathies such as sickle cell disease and β-thalassemia.
T40155 FTX-6058 hydrochloride

FTX-6058 hydrochloride is a potent and orally active inhibitor of Embryonic Ectoderm Development (EED), with the ability to induce HbF protein expression in both cell and murine models. This compound is particularly valuable in the research of select hemoglobinopathies, such as sickle cell disease and β-thalassemia.
T73517 RK-701

RK-701 是一种G9a 高选择性且非遗传毒性的抑制剂,IC50值为 23-27 nM。RK-701 选择性的上调 HbF、γ- Globin、BGLT3 的表达,下调 H3K9me2 的表达。RK-701 也对 BCL11A 和 ZBTB7A 有抑制作用。

化合物

HBF-0259
Cat.No: T27527
Synonym: HBF 0259
Target: Antiviral
HbF inducer-1
Cat.No: T60898
Synonym:
Target:
RN-1 dihydrochloride
Cat.No: T21652
Synonym:
Target: Histone Demethylase, MAO
TN1
Cat.No: T19583
Synonym:
Target: Others
FTX-6058
Cat.No: T40154
Synonym:
Target:
FTX-6058 hydrochloride
Cat.No: T40155
Synonym:
Target:
RK-701
Cat.No: T73517
Synonym:
Target:
TargetMol Loading
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