首页 工具
登录
购物车

搜索结果

Search Results for " hmvec "

2

抑制剂 & 化合物

1

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T4478 CID 16020046

C390-0219

Cannabinoid Receptor GPCR/G Protein
CID 16020046 (C390-0219) 是一种选择性 GPR55 拮抗剂,在酵母中抑制 GPR55 组成型活性,IC50 为 0.15 μM。它抑制 GPR55 介导的 Ca2+信号传导和 GPR55 介导的 ERK1/2 磷酸化,可降低内皮细胞的伤口愈合,参与血小板功能的调节。
T36717 RWJ-56110 dihydrochloride

RWJ-56110 dihydrochloride is a potent, selective, peptide-mimetic inhibitor of PAR-1 activation and internalization (binding IC50=0.44 uM) and shows no effect on PAR-2, PAR-3, or PAR-4. RWJ-56110 dihydrochloride inhibits the aggregation of human platelets induced by both SFLLRN-NH2 (IC50=0.16 μM) and thrombin (IC50=0.34 μM), quite selective relative to U46619 . RWJ-56110 dihydrochloride blocks angiogenesis and blocks the formation of new vessels in vivo. RWJ-56110 dihydrochloride induces cell ap...

化合物

CID 16020046
Cat.No: T4478
Synonym: C390-0219
Target: Cannabinoid Receptor
RWJ-56110 dihydrochloride
Cat.No: T36717
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5S2347 Deoxyshikonin

去氧紫草素,Arnebin 7

Others; HIF/HIF Prolyl-Hydroxylase; Antibacterial Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Others
Deoxyshikonin (Arnebin 7) 是从紫草中分离的天然产物,具有抗肿瘤活性,在体外具有促血管生成作用。它和没食子酸十二烷基酯在体内外均与青霉素有显着的协同抗菌活性。

天然产物

Deoxyshikonin
Cat.No: T5S2347
Synonym: 去氧紫草素,Arnebin 7
Target: Others, HIF/HIF Prolyl-Hydroxylase, Antibacterial
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼