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Cat. No. Product Name Target Signaling Pathways
T32090 HMS-I2

HMSI2,HMS I2

HMS-I2 is a chemical probe used to form heterochromatin. It works by disrupting heterochromatin mediated transcriptional gene silencing.
T32089 HMS-I1 Hydrobromide

HMS-I1 HBr

HMS-I1 Hydrobromide is a probe that works by destroying heterochromatin mediated transcriptional gene silencing and is used for studies of heterochromatin formation and function.
T15159 Dorzagliatin

HMS5552

Glucokinase Metabolism
Dorzagliatin (HMS5552) 是双重作用的葡萄糖激酶 (glucokinase;GK) 激活剂,可改善 2 型糖尿病的血糖控制,提高胰腺 β 细胞功能。
T28781 Sinogliatin

HMS-5552,RO 5305552,HMS5552,RO5305552,HMS 5552,RO-5305552

Sinogliatin, a glucokinase activator, is used potentially for the treatment of type 2 diabetes.
T69365 HMS607P03

HMS607P03 is an activator of SIRT1 which induces autophagic cell death via the AMPK-mTOR-ULK complex and induces mitophagy by the SIRT1-PINK1-Parkin pathway. HMS607P03 downregulates 14-3-3γ, catalase, profilin-1, and HSP90α.
T0977 Medrysone

Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松

Glucocorticoid Receptor; Others Endocrinology/Hormones; Others
Medrysone (6α-Methyl-11β-hydroxyprogesterone) 是局部合成的糖皮质激素,具有代谢、抗炎和抗过敏特性,有潜力用于眼科的眼炎症研究。

化合物

HMS-I2
Cat.No: T32090
Synonym: HMSI2,HMS I2
Target:
HMS-I1 Hydrobromide
Cat.No: T32089
Synonym: HMS-I1 HBr
Target:
Dorzagliatin
Cat.No: T15159
Synonym: HMS5552
Target: Glucokinase
Sinogliatin
Cat.No: T28781
Synonym: HMS-5552,RO 5305552,HMS5552,RO5305552,HMS 5552,RO-5305552
Target:
HMS607P03
Cat.No: T69365
Synonym:
Target:
Medrysone
Cat.No: T0977
Synonym: Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松
Target: Glucocorticoid Receptor, Others
TargetMol Loading
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