Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T36420 |
IM-156 acetate
HL271 acetate |
||
IM-156 acetate 是一种 NADH 脱氢酶(IC50=2.2μM)和 AMP-激活蛋白激酶α(AMPKα)的激活剂,是一种可口服且具有生物利用的线粒体氧化磷酸化(OxPhos)抑制剂。IM-156 acetate 可增加 AMPKα活性,抑制氯己酮诱导的大鼠腹膜纤维化,抑制肿瘤生长 。 | |||
T11570 |
HL271
|
AMPK | Chromatin/Epigenetic; PI3K/Akt/mTOR signaling |
HL271, a derivative of metformin, is a potent AMPK activator that increases AMPK phosphorylation. HL271 attenuates aging-associated cognitive impairment. |