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Cat. No. Product Name Target Signaling Pathways
TN4174 Guajadial

Glucokinase Metabolism
Guajadial shows α-glucosidase inhibitory activities significantly and its activity was better than that of Acarbose.Guajadial may act as Selective Estrogen Receptors Modulators (SERMs), therefore holding significant potential for anticancer therapy, it ex
TN5348 Guajadial F

Guajadial F acts as a Top1 catalytic inhibitor and can delay Top1 poison-mediated DNA damage. Guajadial F shows cytotoxicity against five human cancer cell lines.
TN5347 Guajadial E

Guajadial E shows cytotoxicity against five human cancer cell lines.
TN5349 Guajadial D

Guajadial D shows cytotoxicity against five human cancer cell lines.
TN4172 Guajadial B

Topoisomerase DNA Damage/DNA Repair
Guajadial B acts as a Top1 catalytic inhibitor and delays Top1 poison-mediated DNA damage. Guajadial B shows cytotoxicities against five human cancer cell lines, it is the most effective having an IC50 value of 150 nM toward A549 cells.
TN4173 Guajadial C

Topoisomerase DNA Damage/DNA Repair
Guajadial C acts as a Top1 catalytic inhibitor and can delay Top1 poison-mediated DNA damage. It shows cytotoxicity against five human cancer cell lines.
TN3969 Epiguajadial B

Others Others
Epiguajadial B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3969,CAS号为 1411629-26-9。

天然产物

Guajadial
Cat.No: TN4174
Synonym:
Target: Glucokinase
Guajadial F
Cat.No: TN5348
Synonym:
Target:
Guajadial E
Cat.No: TN5347
Synonym:
Target:
Guajadial D
Cat.No: TN5349
Synonym:
Target:
Guajadial B
Cat.No: TN4172
Synonym:
Target: Topoisomerase
Guajadial C
Cat.No: TN4173
Synonym:
Target: Topoisomerase
Epiguajadial B
Cat.No: TN3969
Synonym:
Target: Others
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