Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11523 |
GZD856
|
PDGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
GZD856 is an orally bioavailable PDGFRα/β inhibitor (IC50s: 68.6 and 136.6 nM) with anti-lung cancer activities. | |||
T64087 | GZD856 formic | ||
GZD856 formic 是一种有效的和具有口服活性的PDGFRα/β抑制剂,IC50值分别为 68.6 和 136.6 nM。GZD856 formic 也是Bcr-AblT315I 的抑制剂,对天然Bcr-Abl 和 T315I 突变型的IC50值分别为 19.9 和 15.4 nM。GZD856 formic 具有抗肿瘤活性。 |