Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6849 |
Uprosertib
GSK2141795,GSK795,优普色替 |
Akt | Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Uprosertib (GSK2141795) 是一种有效的,选择性的 Akt 广谱抑制剂,对 Akt1/Akt2/Akt3 的 IC50值分别为 180/328/38 nM。 | |||
T15428 |
Uprosertib hydrochloride
GSK2141795 (hydrochloride) |
Others | Others |
Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively). |