Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1906 |
Molibresib
GSK 525762A,GSK525762,(4S)-6-(4-氯苯基)-N-乙基-8-甲氧基-1-甲基-4H-[1,2,4]三唑并[4,3-a][1,4]苯并二氮杂卓-4-乙酰胺,I-BET 762 |
Epigenetic Reader Domain | Chromatin/Epigenetic |
Molibresib (GSK525762) 是一种 BET 溴结构域抑制剂,IC50为32.5在42.5 nM 之间。 | |||
T11472L |
Molibresib besylate
I-BET 762 besylate,GSK 525762C |
CCR | Immunology/Inflammation; Microbiology/Virology |
Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM). | |||
T11472 |
GSK 525768A
|
Others | Others |
GSK 525768A, the inactive enantiomer of GSK525762A, exhibits no activity towards BET. |