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Cat. No. Product Name Target Signaling Pathways
T1894 Idelalisib

艾代拉里斯,GS-1101,CAL-101

PI3K; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Idelalisib (GS-1101) 是 PI3K 催化亚基 p110δ 的小分子抑制剂,IC50为 2.5 nM,对 p110δ 的选择性是 p110α/β/γ 的 40 到 300 倍。
T8651 CAL-101

(S)-2-(1-(9H-Purin-6-ylamino)ethyl)-5-fluoro-3-phenylquinazolin-4(3H)-one,GS-1101,Idelalisib

PI3K PI3K/Akt/mTOR signaling
CAL-101 (Idelalisib) 是 p110δ 的选择性抑制剂(IC50:2.5 nM;在无细胞试验中);显示对 p110δ 的选择性比 p110α/β/γ 高 40 到 300 倍,对 p110δ 的选择性比 C2β、hVPS34、DNA-PK 和 mTOR 高 400 到 4000 倍。
T16716 Rabacfosadine

VDC-1101,GS-9219

Others Others
Rabacfosadine is a novel prodrug of the nucleotide analogue PMEG and is designed as a cytotoxic agent.
T24702 Rabacfosadine succinate

VDC-1101 succinate,GS-9219 succinate,VDC 1101 succinate VDC1101 succinate,GS-9219-01

Rabacfosadine succinate is the acyclic nucleoside phosphonate PMEG double prodrug.
T11610 Idelalisib D5

CAL-101 D5,GS-1101 D5

PI3K PI3K/Akt/mTOR signaling
Idelalisib D5 is a deuterium-labeled Idelalisib. Idelalisib is a highly selective and orally bioavailable p110δ inhibitor.

化合物

Idelalisib
Cat.No: T1894
Synonym: 艾代拉里斯,GS-1101,CAL-101
Target: PI3K, Autophagy
CAL-101
Cat.No: T8651
Synonym: (S)-2-(1-(9H-Purin-6-ylamino)ethyl)-5-fluoro-3-phenylquinazolin-4(3H)-one,GS-1101,Idelalisib
Target: PI3K
Rabacfosadine
Cat.No: T16716
Synonym: VDC-1101,GS-9219
Target: Others
Rabacfosadine succinate
Cat.No: T24702
Synonym: VDC-1101 succinate,GS-9219 succinate,VDC 1101 succinate VDC1101 succinate,GS-9219-01
Target:
Idelalisib D5
Cat.No: T11610
Synonym: CAL-101 D5,GS-1101 D5
Target: PI3K
TargetMol Loading
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