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Targets Recommended: GHSR

2

抑制剂 & 化合物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T11560 hGPR91 antagonist 1

(S)-2-(4-(1,8-萘啶-2-基)苯基)-N-(1-(4'-氟-3'-(三氟甲基)-[1,1'-联苯]-4-基)乙基)乙酰胺

GHSR GPCR/G Protein
HGPR91 antagonist 1 是小分子hGPR91选择性拮抗剂(IC50:7 μM)。
T62858 hGPR91 antagonist 3

GPR Endocrinology/Hormones; GPCR/G Protein
hGPR91 antagonist 3 是一种具有口服活性、有效性和选择性的 hGPR91 拮抗剂。hGPR91 antagonist 3 可用于研究高血压、自身免疫性疾病和视网膜血管生成方面的疾病。

化合物

hGPR91 antagonist 1
Cat.No: T11560
Synonym: (S)-2-(4-(1,8-萘啶-2-基)苯基)-N-(1-(4'-氟-3'-(三氟甲基)-[1,1'-联苯]-4-基)乙基)乙酰胺
Target: GHSR
hGPR91 antagonist 3
Cat.No: T62858
Synonym:
Target: GPR
Cat. No. Product Name Species Expression System
TMPH-02612 CXCR3 Protein, Mouse, Recombinant (His & KSI)

CXC-R3,CKR-L2,CXCR3,CD183,GPR9,Interferon-...

Mouse E. coli
Receptor for the C-X-C chemokine CXCL9, CXCL10 and CXCL11 and mediates the proliferation, survival and angiogenic activity of mesangial cells through a heterotrimeric G-protein signaling pathway. Probably promotes cell chemotaxis response. Binds to CCL21.
TMPH-01162 CXCR3 Protein, Human, Recombinant (GST & His)

IP-10 receptor,CXCR3,CXC-R3,GPR9,Interfero...

Human E. coli
CXCR3 Protein, Human, Recombinant (GST & His) is expressed in E. coli.

重组蛋白

CXCR3 Protein, Mouse, Recombinant (His & KSI)
Cat.No: TMPH-02612
Species: Mouse
Expression System: E. coli
CXCR3 Protein, Human, Recombinant (GST & His)
Cat.No: TMPH-01162
Species: Human
Expression System: E. coli
TargetMol Loading
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