2
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11560 |
hGPR91 antagonist 1
(S)-2-(4-(1,8-萘啶-2-基)苯基)-N-(1-(4'-氟-3'-(三氟甲基)-[1,1'-联苯]-4-基)乙基)乙酰胺 |
GHSR | GPCR/G Protein |
HGPR91 antagonist 1 是小分子hGPR91选择性拮抗剂(IC50:7 μM)。 | |||
T62858 |
hGPR91 antagonist 3
|
GPR | Endocrinology/Hormones; GPCR/G Protein |
hGPR91 antagonist 3 是一种具有口服活性、有效性和选择性的 hGPR91 拮抗剂。hGPR91 antagonist 3 可用于研究高血压、自身免疫性疾病和视网膜血管生成方面的疾病。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02612 |
CXCR3 Protein, Mouse, Recombinant (His & KSI)
CXC-R3,CKR-L2,CXCR3,CD183,GPR9,Interferon-... |
Mouse | E. coli |
Receptor for the C-X-C chemokine CXCL9, CXCL10 and CXCL11 and mediates the proliferation, survival and angiogenic activity of mesangial cells through a heterotrimeric G-protein signaling pathway. Probably promotes cell chemotaxis response. Binds to CCL21. | |||
TMPH-01162 |
CXCR3 Protein, Human, Recombinant (GST & His)
IP-10 receptor,CXCR3,CXC-R3,GPR9,Interfero... |
Human | E. coli |
CXCR3 Protein, Human, Recombinant (GST & His) is expressed in E. coli. |