Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T36036 |
CAY10786
GPR52 antagonist-1 |
GPR | Endocrinology/Hormones; GPCR/G Protein |
CAY10786 (GPR52 antagonist-1) 是 G 蛋白偶联受体 52 (GPR52, IC50 = 0.63 μM) 的拮抗剂。 | |||
T78078 |
GPR52 receptor modulator 1
|
Others | Others |
GPR52受体调制剂1(程序1)是一种有潜力用于神经精神疾病研究的GPR52受体调节剂。 | |||
T9452 |
PW0787
|
GPR | Endocrinology/Hormones; GPCR/G Protein |
PW0787 是一种可透过血脑屏障的,口服具有活性的GPR52选择性激动剂 (EC50=135 nM)。它能够抑制精神刺激行为。 | |||
T15352 |
FTBMT
|
GPR | Endocrinology/Hormones; GPCR/G Protein |
FTBMT 是一种选择性的GPR52激动剂(EC50:75 nM),具有抗精神病和促进认知的作用。 | |||
T70993 |
WO-459
|
||
WO-459 is a novel GPR52 agonist, dose-dependently inducing elevation of intracellular cAMP in HEK293/GPR52 cells. |