首页工具

登录

搜索结果

Search Results for " ghsr "

如果没找到您满意的产品或者您对产品有其他要求，可以联系我们专业顾问为您提供针对性的合理建议。 QQ咨询网站留言咨询

Cat. No.	Product Name	Target	Signaling Pathways
T17103	TM-N1324	Others; GHSR	GPCR/G Protein; Others
	TM-N1324 是一种 GPR39 激动剂。 TM-N1324 在没有和存在 Zn2+ 的情况下分别以 280 nM 和 9 nM 的高效率和效力激活人 GPR39。 TM-N1324 对鼠 GPR39 表现出相似的效力，EC50 分别为 180 nM 和 5 nM。
T4648	TC-G-1008 GPR39-C3	GHSR	GPCR/G Protein
	TC-G-1008 (GPR39-C3) 是一种口服有活性的 GPR39激动剂，可作用于大鼠受体(EC50: 0.4 nM)和人类受体(EC50:0.8 nM)的。
TQ0022	Capromorelin Tartrate 卡普瑞林酒石酸盐,CP 424391-18	GHSR	GPCR/G Protein
	Capromorelin Tartrate (CP 424391-18) 是口服有活性的 growth hormone secretagogue receptor 有效激动剂，能够作用于 hGHS-R1a(Ki:7 nM)。
T16508	PF-5190457 PF-05190457	GHSR	GPCR/G Protein
	PF-5190457 是具有选择性的、有效的生长素释放肽受体选择性的反向激动剂(pKi:8.36)。
T10319	Anamorelin RC-1291,阿拉莫林,ONO-7643	GHSR	GPCR/G Protein
	Anamorelin (ONO-7643) 是新型ghrelin receptor 激动剂，根据FLIPR 检测，得到其EC50=0.74 nM。
T7112	Ibutamoren Mesylate MK-0677,伊布莫仑甲磺酸盐,MK-677	GHSR	GPCR/G Protein
	Ibutamoren Mesylate (MK-0677) 是非肽段类生长激素促分泌素受体 (GHSR) 激动剂，也是一种口服有活性的生长激素 (GH) 促分泌素。
T7225	AnaMorelin hydrochloride RC-1291 hydrochloride,阿拉莫林盐酸盐,ONO-7643 hydrochloride	GHSR	GPCR/G Protein
	AnaMorelin hydrochloride (RC-1291 hydrochloride) 是生长素受体激动剂，根据 FLIPR 检测，得到 EC50=0.74 nM。
T34281	Relamorelin BIM28131,RM 131,BIM-28131,BIM-28163,BIM 28163,BIM28163,BIM 28131	GHSR	GPCR/G Protein
	Relamorelin (RM-131)是一种具有选择性和有效性的生长素释放肽/生长激素促分泌素受体 (GHSR) 激动剂，是一种有效的生长素释放肽模拟物，对 GHS-1a 受体具有很高的亲和力。Relamorelin 是一种具有中枢渗透性的五肽，可增加生长激素水平，加速胃排空，具有研究恶病质的潜力。
T31734	BMS-604992 EX1314,EX-1314 HCl,EX-1314,BMS604992,EX-1314 hydrochloride, BMS-604992,EX 1314
	EX-1314 (BMS-604992) is a growth hormone secretagogue receptor (GHSR) agonist.
T38959	BMS-604992 dihydrochloride EX-1314 dihydrochloride,BMS-604992 dihydrochloride
	BMS-604992 (EX-1314) dihydrochloride is a selective and orally active small-molecule agonist of the growth hormone secretagogue receptor (GHSR). It exhibits high-affinity binding (k i = 2.3 nM) and potent functional activity (EC 50 = 0.4 nM). Furthermore, BMS-604992 dihydrochloride has been shown to stimulate food intake in rodents.
T40876	BMS-604992 free base BMS-604992 free base,EX-1314 free base
	BMS-604992 (EX-1314) free base is a selective, orally active small-molecule growth hormone secretagogue receptor (GHSR) agonist. It exhibits high-affinity binding (k i = 2.3 nM) and potent functional activity (EC 50 = 0.4 nM). Moreover, BMS-604992 free base has the ability to stimulate food intake in rodents.
T28812	SM-130686 SM 130686,SM130,686,SM 130,686
	SM-130,686 is a potent, orally-active agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) and growth hormone secretagogue. It has around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.
T68276	Macimorelin acetate EP-1572 acetate ; AEZS-130 acetate,AEZS-130 acetate,EP-1572 acetate
	Macimorelin (EP-1572) acetate，一种 GH 促分泌素，是一种具有口服活性的GHSR 激动剂。Macimorelin acetate 可刺激 GH 的释放。Macimorelin acetate 可用于成人生长激素缺乏症 (AGHD) 和癌症厌食-恶病质综合征 (CACS) 的研究。
T76318	GHRF, porcine
	GHRF, porcine 是一种生长激素释放激素 (GHRH) 多肽 (porcine)。GHRF, porcine 与 GHRHR 受体结合并促进生长激素的释放。
T75262	Relamorelin TFA
	Relamorelin (RM-131) TFA，一种生长素类似物，是一种选择性的生长素释放肽/生长激素促分泌素受体 (GHSR) 激动剂，对GHS-1a 受体的Ki 值为 0.42 nM。Relamorelin TFA 是一种五肽，具有中枢渗透性。Relamorelin TFA 增加生长激素水平，加速胃排空，具有用于恶病质、胃轻瘫和胃/肠运动障碍研究的潜力。
T39236	Relamorelin acetate Relamorelin acetate,RM-131 acetate,BIM-28131acetate
	Relamorelin (RM-131) acetate is a pentapeptide ghrelin analog that acts as a selective agonist for the ghrelin/growth hormone secretagogue receptor (GHSR). It exhibits a high affinity for the GHS-1a receptor, with a Ki value of 0.42 nM. Notably, Relamorelin acetate can cross the blood-brain barrier and target the central nervous system. This compound effectively increases growth hormone levels and promotes faster gastric emptying. Due to these properties, Relamorelin acetate holds promise for it...

化合物

Cat.No: T17103

Target: Others, GHSR

Cat.No: T4648

Synonym: GPR39-C3

Target: GHSR

Capromorelin Tartrate

Cat.No: TQ0022

Synonym: 卡普瑞林酒石酸盐,CP 424391-18

Target: GHSR

Cat.No: T16508

Synonym: PF-05190457

Target: GHSR

Cat.No: T10319

Synonym: RC-1291,阿拉莫林,ONO-7643

Target: GHSR

Ibutamoren Mesylate

Cat.No: T7112

Synonym: MK-0677,伊布莫仑甲磺酸盐,MK-677

Target: GHSR

AnaMorelin hydrochloride

Cat.No: T7225

Synonym: RC-1291 hydrochloride,阿拉莫林盐酸盐,ONO-7643 hydrochloride

Target: GHSR

Cat.No: T34281

Synonym: BIM28131,RM 131,BIM-28131,BIM-28163,BIM 28163,BIM28163,BIM 28131

Target: GHSR

Cat.No: T31734

Synonym: EX1314,EX-1314 HCl,EX-1314,BMS604992,EX-1314 hydrochloride, BMS-604992,EX 1314

BMS-604992 dihydrochloride

Cat.No: T38959

Synonym: EX-1314 dihydrochloride,BMS-604992 dihydrochloride

BMS-604992 free base

Cat.No: T40876

Synonym: BMS-604992 free base,EX-1314 free base

Cat.No: T28812

Synonym: SM 130686,SM130,686,SM 130,686

Macimorelin acetate

Cat.No: T68276

Synonym: EP-1572 acetate ; AEZS-130 acetate,AEZS-130 acetate,EP-1572 acetate

Cat.No: T76318

Relamorelin TFA

Cat.No: T75262

Relamorelin acetate

Cat.No: T39236

Synonym: Relamorelin acetate,RM-131 acetate,BIM-28131acetate

我们的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。

Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved. 沪ICP备20019793号-4

沪公网安备 31010602006700号

沪公网安备 31010602006700号

TargetMol Loading

联系我们

电话：

400-820-0310

邮箱：

service@tsbiochem.com

QQ：

2881945090（终端用户）

2885109491（经销商）

经销：

终端：

地址：

上海市静安区江场三路238号8楼