Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0765 |
Fomepizole
Antizol-Vet,4-甲基吡唑,甲吡唑,4-Methylpyrazole,Antizol |
P450; CAT; AChR | Metabolism; Neuroscience; oxidation-reduction |
Fomepizole (4-Methylpyrazole) 是细胞色素 P450 (CYP2E1) 抑制剂。它是乙醇脱氢酶 (alcohol dehydrogenase) 竞争性抑制剂。它能够阻断甲醇和乙二醇进一步转化为有毒代谢产物。它具有成为乙二醇或甲醇中毒的解毒剂的潜力。 | |||
T72245 |
Fomepizole hydrochloride
4-Methylpyrazole hydrochloride |
||
Fomepizole hydrochloride(4-Methylpyrazole)是一种高效、具口服活性的细胞色素P450(CYP2E1)和竞争性乙醇脱氢酶(alcohol dehydrogenase)抑制剂,阻止甲醇和乙二醇转化为有毒代谢产物,具有用于乙二醇或甲醇中毒解毒的潜力。 |